EC Number   |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
|---|
    4.1.1.7 | 0.36 |
- |
benzoylphosphonate |
prolonged incubation of BFD with benzoylphosphonate results in permanent inactivation of the enzyme |
680368 |
| 4.1.1.7 | 0.38 |
- |
methyl benzoylphosphonate |
- |
702289 |
| 4.1.1.7 | 1 |
- |
(R)-mandelate |
pH 6.5, wild-type enzyme |
654692 |
| 4.1.1.7 | 2 |
5 |
2-oxohexanoic acid |
pH 6.0, 30°C, wild-type enzyme |
666806 |
| 4.1.1.7 | 10 |
- |
2-oxohexanoic acid |
pH 6.0, 30°C, mutant enzyme A460I |
666806 |
| 4.1.1.7 | 20 |
- |
2-oxopentanoic acid |
pH 6.0, 30°C, wild-type enzyme and mutant enzyme A460I |
666806 |
| 4.1.1.7 | 40 |
- |
(R)-mandelate |
pH 6.5, mutant enzyme H281A |
654692 |
| 4.1.1.7 | 40 |
- |
(R)-mandelate |
pH 6.5, mutant enzyme H70A |
654692 |
| 4.1.1.7 | 45 |
- |
benzoylformate |
mutant enzyme L476P |
682628 |
| 4.1.1.7 | 48 |
- |
2-oxo-4-methylhexanoic acid |
pH 6.0, 30°C, mutant enzyme A460I |
666806 |
