EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.6.4.13 | -999 |
- |
more |
inhibition kinetics |
756012 |
3.6.4.13 | 0.007 |
- |
benzoyl-Nle-Lys-Arg-Arg |
full-length enzyme in presence of cofactor CF40-Gly4-Ser-Gly4-NS3FL |
695648 |
3.6.4.13 | 0.097 |
- |
2'-deoxythymidine 5'-phosphoryl-beta,gamma-hypophosphate |
i.e. ppopT, dTTP analogue, inhibition of NTPase activity of NS3 protein by NTP derivatives |
696161 |
3.6.4.13 | 0.109 |
- |
N1-OH-ITP |
inhibition of NTPase activity of NS3 protein by NTP derivatives |
696161 |
3.6.4.13 | 0.116 |
- |
2',3'-ddATP |
inhibition of NTPase activity of NS3 protein by NTP derivatives |
696161 |
3.6.4.13 | 0.116 |
- |
2'-dTTP |
inhibition of NTPase activity of NS3 protein by NTP derivatives |
696161 |
3.6.4.13 | 0.141 |
- |
3'-dATP |
inhibition of NTPase activity of NS3 protein by NTP derivatives |
696161 |
3.6.4.13 | 0.145 |
- |
beta,gamma-methylene-ATP |
efficient inhibitor, like the N1-oxides N1-O-ATP and N1-OH-ITP |
696161 |
3.6.4.13 | 0.2 |
- |
2-amino-ATP |
pH 7.5, 37°C, wild-type enzyme, inhibition of the ATPase reaction |
713144 |
3.6.4.13 | 0.205 |
- |
N1-O-ATP |
inhibition of NTPase activity of NS3 protein by NTP derivatives |
696161 |