EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.5.1.13 | 0.00005 |
- |
N-benzyl-N-dodecyl-N,N-dimethylammonium chloride |
wild type, substrate: m-(acetamido)N,N,N-trimethylanilinium, inhibition depends on substrate concentration |
697867 |
3.5.1.13 | 0.013 |
- |
N-benzyl-N-dodecyl-N,N-dimethylammonium chloride |
mutant D70G, substrate: m-(acetamido)N,N,N-trimethylanilinium |
697867 |
3.5.1.13 | 0.09 |
- |
serotonin |
wild type, substrate: m-(acetamido)N,N,N-trimethylanilinium |
697867 |
3.5.1.13 | 0.2 |
- |
AgNO3 |
- |
696876 |
3.5.1.13 | 0.2 |
- |
HgCl2 |
- |
696876 |
3.5.1.13 | 0.25 |
- |
p-benzoquinone |
- |
208985 |
3.5.1.13 | 0.27 |
- |
serotonin |
mutant D70G, substrate: m-(acetamido)N,N,N-trimethylanilinium |
697867 |
3.5.1.13 | 0.3 |
- |
N-benzyl-N-dodecyl-N,N-dimethylammonium chloride |
value above 0.3 mM, mutant D70G, substrate: o-nitroacetanilide, inhibition depends on substrate concentration |
697867 |
3.5.1.13 | 0.37 |
- |
N-benzyl-N-dodecyl-N,N-dimethylammonium chloride |
wild type, substrate: o-nitroacetanilide |
697867 |
3.5.1.13 | 2.4 |
- |
tyramine |
wild type, substrate: m-(acetamido)N,N,N-trimethylanilinium |
697867 |