EC Number   |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
|---|
   3.4.22.56 | -999 |
- |
more |
inhibition kinetics, first-order inhibition kinetics and two-step irreversible inhibition mechanism |
717272 |
| 3.4.22.56 | -999 |
- |
more |
Ki-value for enzyme from THP.1 cells with the inhibitor Ac-DEVD-aldehyde is below 1 nM |
647618 |
| 3.4.22.56 | 0.00000023 |
- |
acetyl-DEVD-aldehyde |
pH 7.5, 25°C |
647423 |
| 3.4.22.56 | 0.00000052 |
- |
acetyl-DEVD-aldehyde |
pH 7.5 |
647635 |
| 3.4.22.56 | 0.0000012 |
- |
(S)-1-benzyl-5-[1-[2-(phenoxymethyl)pyrrolidinyl]sulfonyl]isatin |
pH 7.5, 30°C |
647598 |
| 3.4.22.56 | 0.0000013 |
- |
Acetyl-Asp-Glu-Val-Asp-aldehyde |
pH 7.5, 22°C |
669888 |
| 3.4.22.56 | 0.0000025 |
- |
5-[[(2S)-2-(phenoxymethyl)pyrrolidin-1-yl]sulfonyl]-1-phenyl-1H-indole-2,3-dione |
Ki-value is calculated from the initial rates |
678321 |
| 3.4.22.56 | 0.0000036 |
- |
N-benxylozycarbonyl-tLeu-Asp |
pH 7.4, 25°C |
696019 |
| 3.4.22.56 | 0.0000065 |
- |
acetyl-Val-Asp-Val-Ala-Asp-aldehyde |
pH 7.5, 22°C |
669888 |
| 3.4.22.56 | 0.000011 |
- |
1-methyl-5-[[(2S)-2-(phenoxymethyl)pyrrolidin-1-yl]sulfonyl]-1H-indole-2,3-dione |
Ki-value is calculated from the initial rates |
678321 |
