EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.4.22.53 | 0.000041 |
- |
Cbz-Leu-DL-Abu-CONH-(CH2)3-morpholine |
in 50 mM Tris-HCl, 50 mM NaCl, 1 mM EDTA, 1 mM EGTA, 0.1% CHAPS, pH 7.5, 10 mM dithiothreitol, 5 mM CaCl2, and less than 5% (v/v) DMSO, temperature not specified in the publication |
717969 |
3.4.22.53 | 0.000068 |
- |
CBZ-Leu-DL-Phe-CONH-(CH2)3-adenin-9-yl |
in 50 mM Tris-HCl, 50 mM NaCl, 1 mM EDTA, 1 mM EGTA, 0.1% CHAPS, pH 7.5, 10 mM dithiothreitol, 5 mM CaCl2, and less than 5% (v/v) DMSO, temperature not specified in the publication |
717969 |
3.4.22.53 | 0.00007 |
- |
Cbz-Leu-DL-Abu-CONH-(CH2)3-adenin-9-yl |
in 50 mM Tris-HCl, 50 mM NaCl, 1 mM EDTA, 1 mM EGTA, 0.1% CHAPS, pH 7.5, 10 mM dithiothreitol, 5 mM CaCl2, and less than 5% (v/v) DMSO, temperature not specified in the publication |
717969 |
3.4.22.53 | 0.000077 |
- |
Cbz-Leu-DL-Abu-CONH-(CH2)3-2-methoxyadenin-9-yl |
in 50 mM Tris-HCl, 50 mM NaCl, 1 mM EDTA, 1 mM EGTA, 0.1% CHAPS, pH 7.5, 10 mM dithiothreitol, 5 mM CaCl2, and less than 5% (v/v) DMSO, temperature not specified in the publication |
717969 |
3.4.22.53 | 0.000209 |
- |
CBZ-Leu-DL-Phe-CONH-(CH2)3-2-methoxyadenin-9-yl |
in 50 mM Tris-HCl, 50 mM NaCl, 1 mM EDTA, 1 mM EGTA, 0.1% CHAPS, pH 7.5, 10 mM dithiothreitol, 5 mM CaCl2, and less than 5% (v/v) DMSO, temperature not specified in the publication |
717969 |
3.4.22.53 | 0.000286 |
- |
Cbz-Leu-DL-Abu-CONH-(CH2)3-(4-methylpiperazin-1-yl) |
in 50 mM Tris-HCl, 50 mM NaCl, 1 mM EDTA, 1 mM EGTA, 0.1% CHAPS, pH 7.5, 10 mM dithiothreitol, 5 mM CaCl2, and less than 5% (v/v) DMSO, temperature not specified in the publication |
717969 |
3.4.22.53 | 0.000438 |
- |
CBZ-Leu-DL-Phe-CONH-(CH2)3-cytosin-3-yl |
in 50 mM Tris-HCl, 50 mM NaCl, 1 mM EDTA, 1 mM EGTA, 0.1% CHAPS, pH 7.5, 10 mM dithiothreitol, 5 mM CaCl2, and less than 5% (v/v) DMSO, temperature not specified in the publication |
717969 |
3.4.22.53 | 0.000844 |
- |
CBZ-Leu-DL-Phe-CONH-(CH2)3-N-(CH3)2 |
in 50 mM Tris-HCl, 50 mM NaCl, 1 mM EDTA, 1 mM EGTA, 0.1% CHAPS, pH 7.5, 10 mM dithiothreitol, 5 mM CaCl2, and less than 5% (v/v) DMSO, temperature not specified in the publication |
717969 |
3.4.22.53 | 0.00092 |
- |
leupeptin |
room temperature, pH 7.5, with succinyl-Met-Leu-methylcoumarin as substrate |
644046 |
3.4.22.53 | 0.00114 |
- |
Cbz-Leu-DL-Abu-CONH-(CH2)3-cytosin-3-yl |
in 50 mM Tris-HCl, 50 mM NaCl, 1 mM EDTA, 1 mM EGTA, 0.1% CHAPS, pH 7.5, 10 mM dithiothreitol, 5 mM CaCl2, and less than 5% (v/v) DMSO, temperature not specified in the publication |
717969 |