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EC Number Ki Value [mM] Ki Value maximum [mM] Inhibitor Commentary Reference
Display the word mapDisplay the reaction diagram Show all sequences 3.4.21.21-999 - more because of competitive binding of p-aminobenzamidine and D-Ile-Pro-Arg-p-nitroanilide, the apparent Ki values were calculated from the p-aminobenzamidine IC50, taking into account the concentration of D-Ile-Pro-Arg-p-nitroanilide ([S]) and the Km for this substrate using Ki =IC50/(1 + [S]/Km) 667474
Display the word mapDisplay the reaction diagram Show all sequences 3.4.21.21-999 - more inhibition kinetics of wild-type and mutant enzymes, overview 683139
Display the word mapDisplay the reaction diagram Show all sequences 3.4.21.210.00000016 - (2R,15R)-2-[(1-aminoisoquinolin-6-yl)amino]-7-(cyclopropanesulfonyl)-4,15,20-trimethyl-13-oxa-4,11-diazatricyclo[14.2.2.16,10]-henicosa-1(18),6,8,10(21),16,19-hexaene-3,12-dione at pH 7.4 and 37°C 754382
Display the word mapDisplay the reaction diagram Show all sequences 3.4.21.210.0000002 - EEWEVLCWTWETCER inhibition of amidolytic activity 654613
Display the word mapDisplay the reaction diagram Show all sequences 3.4.21.210.00000023 - (2R,15R)-2-[(1-amino-7-fluoroisoquinolin-6-yl)amino]-7-(cyclopropanesulfonyl)-4,15,17-trimethyl-13-oxa-4,11-diazatricyclo-[14.2.2.16,10]henicosa-1(18),6,8,10(21),16,19-hexaene-3,12-dione at pH 7.4 and 37°C 754382
Display the word mapDisplay the reaction diagram Show all sequences 3.4.21.210.00000028 - [(2R,15R)-2-[(1-aminoisoquinolin-6-yl)amino]-4,15,20-trimethyl-3,12-dioxo-13-oxa-4,11-diazatricyclo[14.2.2.16,10]henicosa-1-(18),6,8,10(21),16,19-hexaen-7-yl](ethoxy)phosphinic acid at pH 7.4 and 37°C 754382
Display the word mapDisplay the reaction diagram Show all sequences 3.4.21.210.00000035 - R-4-[2-(3-aminobenzenesulfonylamino)-1-(3,5-diethoxy-2-fluorophenyl)-2-oxoethylamino]-2-hydroxy-benzamidine - 669430
Display the word mapDisplay the reaction diagram Show all sequences 3.4.21.210.00000043 - (2R,15R)-2-[(1-amino-4-fluoroisoquinolin-6-yl)amino]-7-(cyclopropanesulfonyl)-4,15,17-trimethyl-13-oxa-4,11-diazatricyclo-[14.2.2.16,10]henicosa-1(18),6,8,10(21),16,19-hexaene-3,12-dione at pH 7.4 and 37°C 754382
Display the word mapDisplay the reaction diagram Show all sequences 3.4.21.210.00000057 - (2R,15R)-2-[(1-aminoisoquinolin-6-yl)amino]-N,N-diethyl-4,15,17-trimethyl-3,12-dioxo-13-oxa-4,11-diazatricyclo[14.2.2.16,10]-henicosa-1(18),6,8,10(21),16,19-hexaene-7-carboxamide at pH 7.4 and 37°C 754382
Display the word mapDisplay the reaction diagram Show all sequences 3.4.21.210.00000061 - diethyl [(2R,15R)-2-[(1-aminoisoquinolin-6-yl)amino]-4,15,17-trimethyl-3,12-dioxo-13-oxa-4,11-diazatricyclo[14.2.2.16,10]henicosa-1(18),6,8,10(21),16,19-hexaen-7-yl]phosphonate at pH 7.4 and 37°C 754382
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