EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.2.1.76 | 0.0012 |
- |
5-fluoro-alpha-L-idopyranosyluronic acid fluoride |
pH 4.5, 37°C |
654716 |
3.2.1.76 | 0.0046 |
- |
2-fluoro-alpha-L-idopyranosyluronic acid fluoride |
pH 4.5, 37°C |
654716 |
3.2.1.76 | 0.094 |
- |
6-sodium-5-amino-5-deoxy-L-idarate-1,5-lactam |
at pH 4.5 and 37°C |
680058 |
3.2.1.76 | 1.3 |
- |
(5S,6R,7S,8S)-5,6,7,8-tetrahydro-6,7,8-trihydroxytetrazolo[1,2-a]pyridine-5-carboxylate |
at pH 4.5 and 37°C |
680058 |
3.2.1.76 | 5 |
- |
(5R,6R,7S,8S)-5,6,7,8-tetrahydro-6,7,8-trihydroxytetrazolo[1,2-a]pyridine-5-carboxylate |
Ki above 5 mM, at pH 4.5 and 37°C |
680058 |
3.2.1.76 | 5 |
- |
(5R,6S,7S,8S)-5,6,7,8-tetrahydro-6,7,8-trihydroxytetrazolo[1,2-a]pyridine-5-carboxylate |
Ki above 5 mM, at pH 4.5 and 37°C |
680058 |
3.2.1.76 | 1831 |
- |
NaCl |
pH 2.8, 37°C, enzyme from healthy individuals |
655246 |