EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
2.8.2.14 | -999 |
- |
more |
inhibition kinetics and modeling, detailed overview |
761727 |
2.8.2.14 | 0.0002 |
- |
adenosine-3',5'-diphosphate |
pH 6.5, 37°C |
645715 |
2.8.2.14 | 0.0002 |
- |
bazedoxifene |
liver cytosol, pH 7.4, 37°C, substrate lithocholic acid, noncompetitive inhibition |
761727 |
2.8.2.14 | 0.0005 |
- |
raloxifene |
liver cytosol, pH 7.4, 37°C, substrate lithocholic acid, noncompetitive inhibition |
761727 |
2.8.2.14 | 0.0006 |
- |
3-ketolithocholate |
pH 6.5, 37°C |
645715 |
2.8.2.14 | 0.0008 |
- |
arzoxifene |
liver cytosol, pH 7.4, 37°C, substrate lithocholic acid, mixed inhibition |
761727 |
2.8.2.14 | 0.0008 |
- |
lasofoxifene |
liver cytosol, pH 7.4, 37°C, substrate lithocholic acid, noncompetitive inhibition |
761727 |
2.8.2.14 | 0.0022 |
- |
glycolithocholate |
pH 6.5, 37°C |
645715 |
2.8.2.14 | 0.0033 |
- |
3-ketolithocholate |
pH 6.5, 37°C |
645717 |
2.8.2.14 | 0.0046 |
- |
droloxifene |
liver cytosol, pH 7.4, 37°C, substrate lithocholic acid, mixed inhibition |
761727 |