EC Number   |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
|---|
    2.7.1.39 | -999 |
- |
more |
- |
641473 |
| 2.7.1.39 | 0.00046 |
- |
4-hydroxy-3-[(4-hydroxy-2-oxo-3,8a-dihydro-2H-chromen-3-yl)methyl]-2H-chromen-2-one |
in 50 mM HEPES, pH 7.5, 40 mM KCl, 10 mM MgCl2, at 37°C |
722043 |
| 2.7.1.39 | 0.0086 |
- |
3-methyl-1-phenyl-6-(trifluoromethyl)-1H-pyrazolo[3,4-b]pyridin-4-ol |
in 50 mM HEPES, pH 7.5, 40 mM KCl, 10 mM MgCl2, at 37°C |
722043 |
| 2.7.1.39 | 0.012 |
- |
(2Z)-2-cyano-N-(2,5-dibromophenyl)-3-hydroxybut-2-enamide |
in 50 mM HEPES, pH 7.5, 40 mM KCl, 10 mM MgCl2, at 37°C |
722043 |
| 2.7.1.39 | 0.0271 |
- |
2-(3,4-dihydroxyphenyl)-3,6,7-trihydroxy-2,3-dihydro-4H-chromen-4-one |
in 50 mM HEPES, pH 7.5, 40 mM KCl, 10 mM MgCl2, at 37°C |
722043 |
| 2.7.1.39 | 0.032 |
- |
1-(naphthalen-2-yl)prop-2-en-1-one |
in 50 mM HEPES, pH 7.5, 40 mM KCl, 10 mM MgCl2, at 37°C |
722043 |
| 2.7.1.39 | 0.0358 |
- |
2-(2-methylpropyl)-6,7,8,9-tetrahydro-4H,5H-cyclohepta[4,5]thieno[2,3-d][1,3]oxazin-4-one |
in 50 mM HEPES, pH 7.5, 40 mM KCl, 10 mM MgCl2, at 37°C |
722043 |
| 2.7.1.39 | 0.1 |
- |
L-homoserine |
in 20% DMSO |
641473 |
| 2.7.1.39 | 0.15 |
- |
L-alpha-aminobutyric acid |
- |
641463 |
| 2.7.1.39 | 0.2 |
0.5 |
(4R)-4-hydroxypentan-2-one |
wild-type enzyme |
641471 |
