EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
2.7.1.32 | -999 |
- |
more |
inhibition kinetics and MIC values |
760133 |
2.7.1.32 | 0.00021 |
- |
hemicholinium-3 |
wild type isoform ChoKalpha1, pH and temperature not specified in the publication |
722672 |
2.7.1.32 | 0.00023 |
- |
hemicholinium-3 |
wild type isoform ChoKalpha2, pH and temperature not specified in the publication |
722672 |
2.7.1.32 | 0.00045 |
- |
hemicholinium-3 |
isoform ChoKalpha2 mutant F352A, pH and temperature not specified in the publication |
722672 |
2.7.1.32 | 0.005 |
- |
hemicholinium-3 |
isoform ChoKbeta mutant F352L, pH and temperature not specified in the publication |
722672 |
2.7.1.32 | 0.008 |
- |
hemicholinium-3 |
isoform ChoKbeta mutant F352A, pH and temperature not specified in the publication |
722672 |
2.7.1.32 | 0.0106 |
- |
1,1'-[[1,1'-biphenyl]-4,4'-diylbis(methylene)]bis[4-[(4-chlorophenyl)(methyl)amino]quinolin-1-ium] |
recombinant enzyme, pH 8.0, 25°C, versus choline |
760133 |
2.7.1.32 | 0.014 |
- |
choline |
pH 8.5, 37°C |
641370 |
2.7.1.32 | 0.016 |
- |
hemicholinium-3 |
isoform ChoKalpha2 mutant F352L, pH and temperature not specified in the publication |
722672 |
2.7.1.32 | 0.0358 |
- |
1,1'-[[1,1'-biphenyl]-4,4'-diylbis(methylene)]bis[4-[(4-chlorophenyl)(methyl)amino]quinolin-1-ium] |
recombinant enzyme, pH 8.0, 25°C, versus ATP |
760133 |