EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
2.5.1.10 | 0.000001 |
- |
1-(2-hydroxy-2,2-diphosphonoethyl)-3-phenylpyridinium |
pH and temperature not specified in the publication |
737349 |
2.5.1.10 | 0.000011 |
- |
zoledronate |
pH and temperature not specified in the publication |
737349 |
2.5.1.10 | 0.00005 |
- |
3-fluoro-1-(2-hydroxy-2,2-diphosphonoethyl)-pyridinium |
pH and temperature not specified in the publication |
737349 |
2.5.1.10 | 0.00026 |
- |
alendronate |
pH and temperature not specified in the publication |
759556 |
2.5.1.10 | 0.000352 |
- |
pamidronate |
pH and temperature not specified in the publication |
759556 |
2.5.1.10 | 0.000388 |
- |
neridronate |
pH and temperature not specified in the publication |
759556 |
2.5.1.10 | 0.00054 |
- |
(R)-(1-((6-(3-chloro-4-methylphenyl)thieno[2,3-d]-pyrimidin-4-yl)amino)-2-(3-fluorophenyl)ethyl)phosphonic acid |
pH 7.7, 37°C |
759612 |
2.5.1.10 | 0.0007 |
- |
isopentenyl diphosphate |
- |
638695 |
2.5.1.10 | 0.001 |
- |
(R)-2-((6-(3-chloro-4-methylphenyl)thieno[2,3-d]-pyrimidin-4-yl)amino)-3-(3-fluorophenyl)propanoic acid |
pH 7.7, 37°C |
759612 |
2.5.1.10 | 0.0011 |
- |
(S)-(1-((6-(3-chloro-4-methylphenyl)thieno[2,3-d]-pyrimidin-4-yl)amino)-2-(3-fluorophenyl)ethyl)phosphonic acid |
pH 7.7, 37°C |
759612 |