EC Number   |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
|---|
   2.1.1.100 | 0.00007 |
- |
sinefungin |
- |
485032 |
| 2.1.1.100 | 0.000296 |
- |
sinefungin |
inhibition of N-acetyl-S-geranylgeranyl-L-cysteinyl-L-alanyl-S-geranylgeranyl-L-cysteine |
485033 |
| 2.1.1.100 | 0.000318 |
- |
sinefungin |
inhibition of N-acetyl-S-(E,E)-farnesyl-L-cysteine methylation |
485033 |
| 2.1.1.100 | 0.0004 |
- |
methyl 3-[[(2E)-5-[4-[2-(biphenyl-4-yl)ethyl]-1H-1,2,3-triazol-1-yl]-3-methylpent-2-en-1-yl]sulfanyl]propanoate |
pH and temperature not specified in the publication |
718467 |
| 2.1.1.100 | 0.0011 |
- |
4-[(naphthalen-2-yl)(thiophen-2-yl)methylidene]oxane |
substrate N-acetyl-S-farnesyl cysteine, pH not specified in the publication, temperature not specified in the publication |
757563 |
| 2.1.1.100 | 0.00117 |
- |
S-Farnesylthioacetic acid |
- |
658348 |
| 2.1.1.100 | 0.0012 |
- |
S-Farnesylthioacetic acid |
- |
485025 |
| 2.1.1.100 | 0.00157 |
- |
S-adenosyl-L-homocysteine |
- |
485032 |
| 2.1.1.100 | 0.0019 |
- |
S-adenosyl-L-homocysteine |
vs. S-adenosyl-L-methionine |
485025 |
| 2.1.1.100 | 0.002 |
- |
S-Farnesylthioacetic acid |
- |
485031 |
