EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
1.14.11.29 | -999 |
- |
more |
inhibition kinetics, overview |
725644 |
1.14.11.29 | -999 |
- |
more |
Ki-values above 0.3 mM: pyridine-2,5-dicarboxylate and 3,4-dihydroxybenzoic acid |
659235 |
1.14.11.29 | 0.0002 |
- |
N-((3-hydroxy-6-chloroquinolin-2-yl)carbonyl)glycine |
pH 7.8, 37°C |
659235 |
1.14.11.29 | 0.0008 |
- |
N-((3-hydroxy-6-chloroquinolin-2-yl)carbonyl)glycine |
pH 7.8, 37°C |
659235 |
1.14.11.29 | 0.001 |
- |
3-hydroxypyridine-2-carbonyl-glycine |
pH 7.8, 37°C |
659235 |
1.14.11.29 | 0.00191 |
- |
3,6,9-tris(naphthalen-1-ylmethyl)-3,6,9,15-tetraazabicyclo[9.3.1]pentadeca-1(15),11,13-triene |
recombinant enzyme, pH 7.0, 37°C |
726084 |
1.14.11.29 | 0.002 |
- |
3-hydroxypyridine-2-carbonyl-glycine |
pH 7.8, 37°C |
659235 |
1.14.11.29 | 0.00249 |
- |
N,N-dimethyl-5-[3,6,9,15-tetraazabicyclo[9.3.1]pentadeca-1(15),11,13-trien-6-ylsulfonyl]naphthalen-1-amine |
recombinant enzyme, pH 7.0, 37°C |
726084 |
1.14.11.29 | 0.00628 |
- |
1,1',1'',1'''-(1,4,7,10-tetraazacyclododecane-1,4,7,10-tetrayl)tetrapropan-2-ol |
recombinant enzyme, pH 7.0, 37°C |
726084 |
1.14.11.29 | 0.007 |
- |
Pyridine-2,4-dicarboxylate |
pH 7.8, 37°C |
659235 |