EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
1.1.1.B40 | 0.000006 |
- |
T0504 |
pH 7.4, 37°C, isozyme 11beta-HSD1, inhibition of cortisol oxidation |
669907 |
1.1.1.B40 | 0.000015 |
- |
T0504 |
pH 7.4, 37°C, isozyme 11beta-HSD1, inhibition of cortisone reduction |
669907 |
1.1.1.B40 | 0.000025 |
- |
T0504 |
pH 7.4, 37°C, isozyme 11beta-HSD1, inhibition of 11-dehydrocorticosterone reduction |
669907 |
1.1.1.B40 | 0.000025 |
- |
T0504 |
pH 7.4, 37°C, isozyme 11beta-HSD1, inhibition of cortisol oxidation |
669907 |
1.1.1.B40 | 0.000028 |
- |
glycyrrhetinic acid |
pH 7.4, 37°C, isozyme 11beta-HSD2, inhibition of cortisol oxidation |
669907 |
1.1.1.B40 | 0.00008 |
- |
T0504 |
pH 7.4, 37°C, isozyme 11beta-HSD1, inhibition of cortisol oxidation |
669907 |
1.1.1.B40 | 0.000082 |
- |
T0504 |
pH 7.4, 37°C, isozyme 11beta-HSD1, inhibition of cortisol oxidation |
669907 |
1.1.1.B40 | 0.00011 |
- |
carbenoxolone |
pH 7.4, 37°C, isozyme 11beta-HSD1, inhibition of cortisol oxidation |
669907 |
1.1.1.B40 | 0.00012 |
- |
glycyrrhetinic acid |
pH 7.4, 37°C, isozyme 11beta-HSD1, inhibition of cortisol oxidation |
669907 |
1.1.1.B40 | 0.00023 |
- |
carbenoxolone |
pH 7.4, 37°C, isozyme 11beta-HSD1, inhibition of 11-dehydrocorticosterone reduction |
669907 |