EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
2.7.4.9 | 0.0058 |
- |
(+/-)(Z)-5-acetamido-1-(4-(thymin-1-yl)but-2-enyl)-5,6-dihydro-1H-imidazo[4,5,1-ij]quinolin-2(4H)-one |
in 50 mM Tris-HCl pH 7.4, 50 mM KCl, 2 mM MgCl2, temperature not specified in the publication |
722186 |
2.7.4.9 | 0.00707 |
- |
(+/-)(Z)-5-amino-1-(4-(thymin-1-yl)but-2-enyl)-5,6-dihydro-1H-imidazo[4,5,1-ij]quinolin-2(4H)-one |
in 50 mM Tris-HCl pH 7.4, 50 mM KCl, 2 mM MgCl2, temperature not specified in the publication |
722186 |
2.7.4.9 | 0.039 |
- |
(3E)-4-[4-[(5-methyl-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)methyl]phenyl]but-3-enoic acid |
- |
691226 |
2.7.4.9 | 0.252 |
- |
(3E)-4-[4-[(5-methyl-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)methyl]phenyl]but-3-enoic acid |
- |
691226 |
2.7.4.9 | 0.0108 |
- |
(4E)-1-(4-hydroxy-3-methoxyphenyl)dec-4-en-3-one |
pH 7.4, temperature not specified in the publication |
738163 |
2.7.4.9 | 0.5 |
- |
(E)-5-(2-bromovinyl)-deoxyuridine |
- |
706485 |
2.7.4.9 | 0.00042 |
- |
(Z)-1-(4-(thymin-1-yl)but-2-enyl)-1H-benzo[c,d]indol-2(1H)one |
pH 7.4 |
691813 |
2.7.4.9 | 0.00116 |
- |
(Z)-1-(4-(thymin-1-yl)but-2-enyl)-5,6-dihydro-1H-imidazo[4,5,1-ij]quinolin-2(4H)-one |
in 50 mM Tris-HCl pH 7.4, 50 mM KCl, 2 mM MgCl2, temperature not specified in the publication |
722186 |
2.7.4.9 | 0.0011 |
- |
(Z)-2-(4-(5-bromouracil-1-yl)but-2-enyl)-1H-benzo[d,e] isoquinoline-1,3(2H)-dione |
pH 7.4 |
691813 |
2.7.4.9 | 0.0019 |
- |
(Z)-2-(4-(thymin-1-yl)but-2-enyl)-1H-benzo[d,e]isoquinoline-1,3(2H)-dione |
pH 7.4 |
691813 |