EC Number   |
Ki Value [mM]   |
Ki Value maximum [mM]   |
Inhibitor   |
Reference   |
|---|
  2.4.2.17 | 0.0811 |
- |
histidine |
25°C, pH 8 |
678174 |
  2.4.2.17 | 1.44 |
- |
AMP |
25°C, pH 8 |
678174 |
  2.4.2.17 | 0.002 |
- |
1-[(5,6-diphenyl-1,2,4-triazin-3-yl)sulfanyl]-3-(1,3-thiazol-2-yl)propan-2-one |
- |
705015 |
  2.4.2.17 | 0.002 |
- |
N-[3-[(6-nitro-1,3-benzothiazol-2-yl)amino]-3-oxo-1-phenylpropyl]benzamide |
- |
705015 |
  2.4.2.17 | 0.004 |
- |
L-histidine |
uncompetitive versus ATP, pH 8.0, 25°C |
721673 |
  2.4.2.17 | 0.0079 |
- |
L-histidine |
uncompetitive versus ATP, pH 8.25, 25°C |
721673 |
  2.4.2.17 | 0.0235 |
- |
L-histidine |
Kii-value, non competitive versus 5-phospho-alpha-D-ribosyl diphosphate, pH 8.5, 25°C |
721673 |
  2.4.2.17 | 0.0257 |
- |
L-histidine |
Kis-value, non competitive versus 5-phospho-alpha-D-ribosyl diphosphate, pH 8.5, 25°C |
721673 |
  2.4.2.17 | 0.0269 |
- |
L-histidine |
uncompetitive versus ATP, pH 8.75, 25°C |
721673 |
  2.4.2.17 | 0.0279 |
- |
L-histidine |
uncompetitive versus ATP, pH 8.5, 25°C |
721673 |