EC Number   |
Ki Value [mM]   |
Ki Value maximum [mM]   |
Inhibitor   |
Reference   |
|---|
  2.4.2.17 | 0.002 |
- |
1-[(5,6-diphenyl-1,2,4-triazin-3-yl)sulfanyl]-3-(1,3-thiazol-2-yl)propan-2-one |
- |
705015 |
  2.4.2.17 | 0.88 |
- |
ADP |
wild type protein, pH 8.5, temperature not specified in the publication |
721765 |
  2.4.2.17 | 0.356 |
- |
AMP |
with respect to ATP, at pH 8.5 and 25°C |
737208 |
  2.4.2.17 | 0.382 |
- |
AMP |
with respect to 5-phospho-alpha-D-ribose 1-diphosphate, at pH 8.5 and 25°C |
737208 |
  2.4.2.17 | 1.29 |
- |
AMP |
wild type protein, pH 8.5, temperature not specified in the publication |
721765 |
  2.4.2.17 | 1.44 |
- |
AMP |
25°C, pH 8 |
678174 |
  2.4.2.17 | 0.0811 |
- |
histidine |
25°C, pH 8 |
678174 |
  2.4.2.17 | 0.0005 |
- |
L-histidine |
wild type enzyme, at pH 8.5 and 30°C |
736541 |
  2.4.2.17 | 0.004 |
- |
L-histidine |
uncompetitive versus ATP, pH 8.0, 25°C |
721673 |
  2.4.2.17 | 0.0079 |
- |
L-histidine |
uncompetitive versus ATP, pH 8.25, 25°C |
721673 |