EC Number |
KM Value [mM] |
KM Value Maximum [mM] |
Substrate |
Reference |
---|
3.5.1.98 | 0.03 |
- |
Ac-Leu-Gly-Lys(Ac)-7-amido-4-methylcoumarin |
apparent KM |
699458 |
3.5.1.98 | 0.0024 |
- |
Fluor de Lys |
catalytic domain II, pH 7.2, 23°C |
677911 |
3.5.1.98 | 1 |
- |
Fluor de Lys HDAC8 substrate |
Co2+-D101A mutant, larger than 1.00 |
696240 |
3.5.1.98 | 0.14 |
- |
Fluor de Lys HDAC8 substrate |
Co2+-D101E mutant |
696240 |
3.5.1.98 | 1 |
- |
Fluor de Lys HDAC8 substrate |
Co2+-D101L mutant, larger than 1.00 |
696240 |
3.5.1.98 | 1 |
- |
Fluor de Lys HDAC8 substrate |
Co2+-D101N mutant, larger than 1.00 |
696240 |
3.5.1.98 | 1 |
- |
Fluor de Lys HDAC8 substrate |
Co2+-H143A mutant, larger than 1.00 |
696240 |
3.5.1.98 | 0.16 |
- |
Fluor de Lys HDAC8 substrate |
Co2+-wild type |
696240 |
3.5.1.98 | -999 |
- |
more |
enzyme kinetic calculations, overview |
733081 |
3.5.1.98 | 0.0054 |
- |
Ac-KGK(acetyl)-7-amido-4-methylcoumarin |
isoform FB188 HDAH |
677964 |