EC Number |
KM Value [mM] |
KM Value Maximum [mM] |
Substrate |
Reference |
---|
3.5.1.98 | 0.0038 |
- |
Fluor de Lys |
mutant H216A, pH 7.2, 23°C |
677911 |
3.5.1.98 | 0.00405 |
- |
Ac-GSK(acetyl)-7-amido-4-methylcoumarin |
isoform HDAC3 |
677964 |
3.5.1.98 | 0.0043 |
- |
Ac-GGK(acetyl)-7-amido-4-methylcoumarin |
isoform HDAC6 |
677964 |
3.5.1.98 | 0.0044 |
- |
Ac-KYK(acetyl)-7-amido-4-methylcoumarin |
isoform HDAC8 |
677964 |
3.5.1.98 | 0.0046 |
- |
Ac-FEK(acetyl)-7-amido-4-methylcoumarin |
isoform HDAC3 |
677964 |
3.5.1.98 | 0.005 |
- |
Ac-KWK(acetyl)-7-amido-4-methylcoumarin |
isoform HDAC1 |
677964 |
3.5.1.98 | 0.0054 |
- |
Ac-KGK(acetyl)-7-amido-4-methylcoumarin |
isoform FB188 HDAH |
677964 |
3.5.1.98 | 0.0056 |
- |
Ac-KYK(acetyl)-7-amido-4-methylcoumarin |
isoform HDAC1 |
677964 |
3.5.1.98 | 0.0056 |
- |
TYSRGGK(Ac)FFRRFP |
pH 7.4, 37°C, recombinant enzyme |
756690 |
3.5.1.98 | 0.00625 |
- |
Ac-IHK(acetyl)-7-amido-4-methylcoumarin |
isoform HDAC6 |
677964 |