EC Number |
Inhibitors |
Structure |
---|
3.4.21.102 | (5S)-SB 214357 |
penem inhibitor, 1 mM, complete loss of activity |
|
3.4.21.102 | CuSO4 |
- |
|
3.4.21.102 | FeCl3 |
- |
|
3.4.21.102 | iodoacetamide |
10 mM, 27% inhibition |
|
3.4.21.102 | more |
insensitive to penem; not inhibitory: phenylmethylsulfonyl fluoride, diisopropyl fluorophosphate, chymostatin, penem, pepstatin A, 2-mercaptoethanol, N-ethylmaleimide, EDTA, 1,10-phenanthroline |
|
3.4.21.102 | more |
insensitive to leupeptin, Nalpha-p-tosyl-L-Lys chloromethyl ketone, 1,10-phenanthroline |
|
3.4.21.102 | more |
oligopeptides with 24 residues corresponding to the substrate with replacements of Asp342 |
|
3.4.21.102 | more |
not inhibitory: EDTA, EGTA, leupeptin, phenylmethylsulfonyl fluoride, iodoacetic acid |
|
3.4.21.102 | more |
complex inhibitors belonging to the substance classes rhodanine dimer, ketoheterocycles, CF3 peptides, and imidazoles were studied, application of inhibitors to the leaves of Arabidopsis thaliana causes lesions, over expression of CtpA results in enhanced resistance to inhibitor treatment |
|
3.4.21.102 | phenylmethylsulfonyl fluoride |
2 mM, 15% inhibition |
|