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Results 1 - 10 of 116 > >>
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EC Number Inhibitors Commentary Structure
Display the word mapDisplay the reaction diagram Show all sequences 2.7.11.12(9S,10R,12R)-2,3,9,10,11,12-hexahydro-10-methoxy-2,9-dimethyl-1-oxo-9,12-epoxy-1H-diindolo [1,2,3-fg:',2',1'-kl]pyrrolo [3,4-i][1,6]benzodiazocine-10-carboxylic acid methyl ester KT-5823, specific PKG inhibitor Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 2.7.11.12(Z)-1-(N-(2-aminoethyl)-N-(2-ammonioethyl)amino)diazen-1-ium-1,2-diolate 24 h exposure to 1 mM (Z)-1-(N-(2-aminoethyl)-N-(2-ammonioethyl)amino)diazen-1-ium-1,2-diolate leads to both reduction in cGKI expression and specific activity Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 2.7.11.121H-[1,2,4]oxadiazolo-[4,3-a]quinoxalin-1-one - Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 2.7.11.122,2'-(hydroxynitrosohydrazono)-bis-ethanamine 24 h incubation with 2,2'-(hydroxynitrosohydrazono)-bis-ethanamine after incubation with cGMP is associated with decreased PKG activity Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 2.7.11.124-methoxy-3,6-diphenylcyclohexa-3,5-diene-1,2-dione isolated from a microbial extract of a Phoma sp. Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 2.7.11.124-[2-(4-fluorophenyl)-5-(1-methylpiperidin-4-yl)-1H-pyrrol-3-yl]pyridine a synthetic compound Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 2.7.11.124-[2-(4-fluorophenyl)-5-(1-methylpiperidine-4-yl)-1H-pyrrol-3-yl]pyridine inhibits downstream of calcium-dependent events, inhibition is not reversible by calcium ionophores or ethanol, inhibits uracil uptake, blocks the attachment of the sporozoite to the host cells and inhibits parasite invasion and gliding motility, inhibits the secretion of micronemal adhesins MIC1 and MIC2 by the parasite, no inhibition of mutants T770M and T770Q Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 2.7.11.124-[2-(4-fluorophenyl)-5-(1-methylpiperidine-4-yl)-1H-pyrrol-3-yl]pyridine inhibits downstream of calcium-dependent events, inhibition is not reversible by calcium ionophores or ethanol, inhibits uracil uptake, blocks the attachment of the tachyzoite to the host cells and inhibits parasite invasion and gliding motility, inhibits the secretion of micronemal adhesin MIC2 by the parasite, no inhibition of mutants T761M and T761Q Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 2.7.11.124-[2-(4-fluorophenyl)imidazo[1,2-a]pyridin-3-yl]-N-[4-(4-methylpiperazin-1-yl)phenyl]pyrimidin-2-amine - Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 2.7.11.124-[2-(4-fluorophenyl)imidazo[1,2-a]pyridin-3-yl]-N-[4-(piperazin-1-yl)phenyl]pyrimidin-2-amine - Go to the Ligand Summary Page
Results 1 - 10 of 116 > >>
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