EC Number |
Inhibitors |
Structure |
---|
1.3.1.22 | (+)-methysticin |
- |
|
1.3.1.22 | (+/-)-LY191704 |
i.e. (4aS,10aR)-7-chloro-1-methyl-3,4,4a,9,10,10a-hexahydrophenanthren-2(1H)-one, non-steroidal, most potent benzoquinoline mimicing 4-azasteroid inhibitors, and specific for isozyme 5alphaR-1, IC50 is 30 nM |
|
1.3.1.22 | (-)-epigallocatechin-3-gallate |
i.e. EGCG, from Thea sativa, slightly inhibits the liver microsomal enzyme |
|
1.3.1.22 | (10bR)-8-chloro-4,10b-dimethyl-4a,5,6,10b-tetrahydrophenanthridin-2(1H)-one |
isoform II, 49% inhibition at 0.02 mM |
|
1.3.1.22 | (10bR)-8-chloro-4,5,10b-trimethyl-4a,5,6,10b-tetrahydrophenanthridin-2(1H)-one |
isoform II, 57% inhibition at 0.029 mM |
|
1.3.1.22 | (10bR)-8-chloro-5,10b-dimethyl-4a,5,6,10b-tetrahydrophenanthridin-2(1H)-one |
isoform II, 42% inhibition at 0.03 mM |
|
1.3.1.22 | (1E,4E,6E)-1,7-bis(3-hydroxy-4-methoxyphenyl)hepta-1,4,6-trien-3-one |
- |
|
1.3.1.22 | (1E,4E,6E)-1,7-bis(3-hydroxyphenyl)hepta-1,4,6-trien-3-one |
- |
|
1.3.1.22 | (1E,4E,6E)-1,7-bis(4-hydroxy-3-methoxyphenyl)hepta-1,4,6-trien-3-one |
- |
|
1.3.1.22 | (1E,4E,6E)-1,7-bis(4-hydroxyphenyl)hepta-1,4,6-trien-3-one |
- |
|