2.1.1.13 0.0014 - ZL-033 at 37°C 684467 2.1.1.13 0.00415 - N-(3-bromo-4-[[(1-[2-[(2,2-dimethylpropanoyl)amino]-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl]aziridin-2-yl)methyl](methyl)amino]benzoyl)-L-glutamic acid pH 7.2, 37°C 733653 2.1.1.13 0.009 - 4-(7-nitroquinoxalin-2-yl)benzoic acid pH 7.4, 37°C 733507 2.1.1.13 0.01 - ZL-031 at 37°C 684467 2.1.1.13 0.018 - 4-nitro-N-[2-(5-nitro-1H-benzimidazol-2-yl)ethyl]benzamide pH 7.4, 37°C 733507 2.1.1.13 0.02 - N-[(5-nitro-1H-benzimidazol-2-yl)methyl]benzamide pH 7.4, 37°C 733507 2.1.1.13 0.08 - 4-nitro-2,1,3-benzothiadiazole IC50: 0.08 mM 673596 2.1.1.13 0.095 - 5-amino-7-methoxy-N1-methylbenzimidazole IC50: 0.095 mM 673596 2.1.1.13 0.1 - 5-nitro-7-methoxybenzimidazole IC50: 0.1 mM 673596 2.1.1.13 0.12 - 2-nitro-1H-benzimidazole IC50: 0.12 mM 673596