2.5.1.21 0.00000051 - 2-(1-[2-[(4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]ethyl]-1H-1,2,3-triazol-4-yl)acetic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.00000059 - 1-[2-[(4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]ethyl]-1H-1,2,3-triazole-4-carboxylic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.00000068 - 2-[(1-[2-[(4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]ethyl]-1H-1,2,3-triazol-4-yl)methoxy]acetic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.00000069 - 2-[(1-[2-[(4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]ethyl]-1H-1,2,3-triazol-4-yl)methoxy]-2-methylpropanoic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.0000007 - zaragozic acid IC50 0.7 nM 489849 2.5.1.21 0.0000008 - 2-[(1-[3-[(4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]propanoyl]-4-piperidinyl)oxy]acetic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.00000081 - 2-(1-[2-[(4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]ethyl]-1H-1,2,3-triazol-5-yl)acetic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.00000084 - E5700 IC50: 0.84 nM 671377 2.5.1.21 0.00000085 - 3-(2-[2-[(4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]ethyl]-2H-1,2,3,4-tetrazol-5-yl)propanoic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.00000089 - 2-[2-[(4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]ethyl]-2H-1,2,3,4-tetrazol-5-carboxylic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.0000009 - 2-[(1-[3-[(4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]propanoyl]-4-piperidinyl)methoxy]acetic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.0000011 - 2-(2-[2-[(4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl)ethyl]-2H-1,2,3,4-tetrazol-5-yl]-2-methylpropanoic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.0000011 - 2-(2-[2-[(4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl)ethyl]-2H-1,2,3,4-tetrazol-5-yl]acetic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.0000011 - 2-(2-[2-[(4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]ethyl]-1H-1,2,3,4-tetrazol-5-yl)acetic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.0000013 - 2-(1-[2-[(4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]acetyl]-4-piperidinyl)acetic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.0000013 - 2-(1-[2-[(4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]ethyl]-1H-pyrazol-3-yl)acetic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.0000014 - (3S)-1-(3-((4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl)propanoyl)-3-piperidine carboxylic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.0000014 - 3-[(1-[3-[(4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]propanoyl]-4-piperidinyl)oxy]propanoic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.0000016 - 2-(1-[2-[(4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]ethyl]-1H-pyrazol-5-yl)acetic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.0000016 - 2-[1,8-dichloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]acetic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.0000016 - 4-[3-[(4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]propanoyl]-2-morpholine carboxylic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.0000017 - 1-(2-[2-[(4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]ethyl]-2H-1,2,3,4-tetrazol-5-yl)cyclopropanecarboxylic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.0000017 - 2-[(1-[2-[(4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]ethyl]-1H-1,2,3-triazol-4-yl)methoxy]-2-ethylbutanoic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.0000021 - 1-[2-[(4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]ethyl]-1H-pyrazole-4-carboxylic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.0000022 - 1-(3-((4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl)propanoyl)-3-azetidine carboxylic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.0000022 - 2-(4-[3-[(4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]propanoyl]-2-oxo-1-piperazinyl)acetic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.0000023 - (3S)-1-[2-[(4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]acetyl]-3-piperidinecarboxylic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.0000023 - 2-([2-[(4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]acetyl]amino)acetic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.0000024 - 2-(1-[3-[(4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]propanoyl]-4-piperidinyl)acetic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.0000025 - 2-[(2-[2-[(4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]ethyl]-2H-1,2,3,4-tetrazol-5-yl)methoxy]-2-methylpropanoic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.0000027 - 2-(1-[2-[8-chloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]acetyl]-4-piperidinyl)acetic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.0000029 - 3-([2-[(4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]acetyl]amino)propionic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.0000031 - 2-(1-[2-[(4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]ethyl]-1H-pyrazol-4-yl)acetic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.0000031 - 3-[(4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-4H,6Hpyrrolo[1,2-a][4,1]benzoxazepin-4-yl]propionic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.0000033 - 2-[8-chloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]acetic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.0000034 - 1-[2-[(4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]acetyl]-4-piperidinecarboxylic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.00000352 - ER119884 IC50: 3.52 nM 671377 2.5.1.21 0.000004 - 3-([2-[(4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]acetyl]amino)benzoic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.0000043 - 2-(4-[2-[(4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]acetyl]-1-piperazinyl)acetic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.000007 - 2-(1-(3-[(4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]propanoyl)-3-azetidinyl)acetic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.0000076 - 2-[8-chloro-6-(2,3-dimethoxyphenyl)-1-(4-morpholinylmethyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]acetic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.00002 - CP-295697 a bisphosphonate, IC50: 20 nM 489849 2.5.1.21 0.00005 - ethyl 4-(1-azabicyclo[2.2.2]oct-2-en-3-yl)benzoate IC50: 50 nM 671377 2.5.1.21 0.000052 - 2-[8-chloro-6-(2,3-dichlorobenzoyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]acetic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.000056 - [(4R,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-1-(propan-2-yl)-6,10b-dihydro-1H,4H-[2]benzoxepino[4,5-c][1,2]oxazol-4-yl]acetic acid pH and temperature not specified in the publication 721802 2.5.1.21 0.0000955 - zaragozic acid A pH 7.2, 37°C 687416 2.5.1.21 0.0001 - chlorogenic acid pH 7.4, 37°C 688316 2.5.1.21 0.000112 - 1-[[(6S)-8-chloro-6-(2,3-dimethoxyphenyl)-1-(propan-2-yl)-6,10b-dihydro-1H,4H-[2]benzoxepino[4,5-c][1,2]oxazol-4-yl]acetyl]piperidine-4-carboxylic acid pH and temperature not specified in the publication 721802 2.5.1.21 0.00013 - CP-294838 a benzoxazepinone IC50 130 nM 489849 2.5.1.21 0.000131 - (1-[[(6S)-8-chloro-6-(2,3-dimethoxyphenyl)-1-(propan-2-yl)-6,10b-dihydro-1H,4H-[2]benzoxepino[4,5-c][1,2]oxazol-4-yl]acetyl]piperidin-4-yl)acetic acid pH and temperature not specified in the publication 721802 2.5.1.21 0.000162 - 2-[(6S)-8-chloro-6-(2,3-dimethoxyphenyl)-1-(propan-2-yl)-6,10b-dihydro-1H,4H-[2]benzoxepino[4,5-c][1,2]oxazol-4-yl]-1-[(3R)-3-hydroxypyrrolidin-1-yl]ethanone pH and temperature not specified in the publication 721802 2.5.1.21 0.000169 - [(4S,6R)-8-chloro-6-(2,3-dimethoxyphenyl)-1-(propan-2-yl)-6,10b-dihydro-1H,4H-[2]benzoxepino[4,5-c][1,2]oxazol-4-yl]acetic acid pH and temperature not specified in the publication 721802 2.5.1.21 0.000213 - (1-[[(3R,5S)-1-[3-(acetyloxy)-2,2-dimethylpropyl]-7-chloro-5-(2,3-dimethoxyphenyl)-2-oxo-1,2,3,5-tetrahydro-4,1-benzoxazepin-3-yl]acetyl]piperidin-4-yl)acetic acid pH and temperature not specified in the publication 721802 2.5.1.21 0.00022 - 1-[[(1R,5R)-7-chloro-5-(2,3-dimethoxyphenyl)-1-(2-methylpropyl)-2-oxo-1,2,4,5-tetrahydro-3H-3-benzazepin-3-yl]acetyl]piperidine-4-carboxylic acid pH and temperature not specified in the publication 721801 2.5.1.21 0.00022 - methyl 2-[8-chloro-6-(2,3-dimethoxyphenyl)-4H,6Hpyrrolo[1,2-a][4,1]benzoxazepin-4-yl]acetate pH 7.2-7.5, 37°C 721838 2.5.1.21 0.000223 - [(6S)-8-chloro-6-(2,3-dimethoxyphenyl)-1-(propan-2-yl)-6,10b-dihydro-1H,4H-[2]benzoxepino[4,5-c][1,2]oxazol-4-yl]acetic acid pH and temperature not specified in the publication 721802 2.5.1.21 0.00026 - (1-[[(3R,5S)-7-chloro-5-(2,3-dimethoxyphenyl)-1-(3-hydroxy-2,2-dimethylpropyl)-2-oxo-1,2,3,5-tetrahydro-4,1-benzoxazepin-3-yl]acetyl]piperidin-4-yl)acetic acid pH and temperature not specified in the publication 721802 2.5.1.21 0.00037 - (1R,5S)-7-chloro-5-(2-methoxyphenyl)-1-(2-methylpropyl)-3-[2-oxo-2-(piperidin-1-yl)ethyl]-1,3,4,5-tetrahydro-2H-3-benzazepin-2-one pH and temperature not specified in the publication 721801 2.5.1.21 0.00044 - 2-[8-chloro-6-(2,3-dihydro-1,4-benzodioxin-5-yl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]acetic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.00045 - 1-[[(1R,5S)-7-chloro-5-(2,3-dimethoxyphenyl)-1-(2-methylpropyl)-2-oxo-1,2,4,5-tetrahydro-3H-3-benzazepin-3-yl]acetyl]piperidine-4-carboxylic acid pH and temperature not specified in the publication 721801 2.5.1.21 0.0005 - 1-[[(1R,5S)-7-chloro-5-(2-methoxyphenyl)-1-(2-methylpropyl)-2-oxo-1,2,4,5-tetrahydro-3H-3-benzazepin-3-yl]acetyl]piperidine-4-carboxylic acid pH and temperature not specified in the publication 721801 2.5.1.21 0.00054 - 2-[8-chloro-6-(2,3-dimethoxyphenyl)-1-[(dimethylamino)methyl]-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]acetic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.0006 - 2-(1-[2-[(4S,6R)-8-chloro-6-(2,3-dimethoxyphenyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]acetyl]-4-piperidinyl)acetic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.0006 - 2-[8-chloro-6-(1-naphthyl)-4H,6H-pyrrolo[1,2-a][4,1]benzoxazepin-4-yl]acetic acid pH 7.2-7.5, 37°C 721838 2.5.1.21 0.00073 - 3-(biphenyl-4-ylmethyl)-1-azabicyclo[2.2.2]oct-2-ene IC50: 730 nM 671377 2.5.1.21 0.00083 - 3-[[4-(benzyloxy)phenyl]ethynyl]-1-azabicyclo[2.2.2]oct-2-ene IC50: 830 nM 671377 2.5.1.21 0.00083 - celastrol pH 7.4, temperature not specified in the publication 758735 2.5.1.21 0.00093 - 1-[[(1R,5S)-7-chloro-5-(2-chlorophenyl)-1-(2-methylpropyl)-2-oxo-1,2,4,5-tetrahydro-3H-3-benzazepin-3-yl]acetyl]piperidine-4-carboxylic acid pH and temperature not specified in the publication 721801 2.5.1.21 0.0012 - [(1R,5S)-7-chloro-5-(2,3-dimethoxyphenyl)-1-(2-methylpropyl)-2-oxo-1,2,4,5-tetrahydro-3H-3-benzazepin-3-yl]acetic acid pH and temperature not specified in the publication 721801 2.5.1.21 0.0014 - (1-[[(1R,5S)-7-chloro-5-(2-chlorophenyl)-1-(2-methylpropyl)-2-oxo-1,2,4,5-tetrahydro-3H-3-benzazepin-3-yl]acetyl]piperidin-4-yl)acetic acid pH and temperature not specified in the publication 721801 2.5.1.21 0.00142 - [(4R,6R)-8-chloro-6-(2,3-dimethoxyphenyl)-1-(propan-2-yl)-6,10b-dihydro-1H,4H-[2]benzoxepino[4,5-c][1,2]oxazol-4-yl]acetic acid pH and temperature not specified in the publication 721802 2.5.1.21 0.0015 - (3R)-3-[[3-(benzyloxy)phenyl]ethynyl]-1-azabicyclo[2.2.2]octan-3-ol IC50: 1500 nM 671377 2.5.1.21 0.0019 - [(1R,5S)-7-chloro-5-(2-methoxyphenyl)-1-(2-methylpropyl)-2-oxo-1,2,4,5-tetrahydro-3H-3-benzazepin-3-yl]acetic acid pH and temperature not specified in the publication 721801 2.5.1.21 0.0022 - [(1R,5S)-5-(2-bromophenyl)-7-chloro-1-(2-methylpropyl)-2-oxo-1,2,4,5-tetrahydro-3H-3-benzazepin-3-yl]acetic acid pH and temperature not specified in the publication 721801 2.5.1.21 0.0024 - 6-([[(1R,5S)-7-chloro-5-(2-chlorophenyl)-1-(2-methylpropyl)-2-oxo-1,2,4,5-tetrahydro-3H-3-benzazepin-3-yl]acetyl]amino)hexanoic acid pH and temperature not specified in the publication 721801 2.5.1.21 0.0033 - [(1R,5S)-7-chloro-5-(2-chlorophenyl)-1-(2-methylpropyl)-2-oxo-1,2,4,5-tetrahydro-3H-3-benzazepin-3-yl]acetic acid pH and temperature not specified in the publication 721801 2.5.1.21 0.0055 - (2E)-3-[(1R,5S)-3-(carboxymethyl)-7-chloro-5-(2-chlorophenyl)-2-oxo-2,3,4,5-tetrahydro-1H-3-benzazepin-1-yl]-2-methylprop-2-enoic acid pH and temperature not specified in the publication 721801 2.5.1.21 0.0055 - [(4S,6S)-8-chloro-6-(2,3-dimethoxyphenyl)-1-(propan-2-yl)-6,10b-dihydro-1H,4H-[2]benzoxepino[4,5-c][1,2]oxazol-4-yl]acetic acid pH and temperature not specified in the publication 721802 2.5.1.21 0.0065 - 4-methyl-2-(3',5'-di-tert-butyl-4'-hydroxy-4-biphenyl)-3,4-dihydro-2H-1,4-benzothiazine-2-ol pH and temperature not specified in the publication 759144 2.5.1.21 0.007 - 2-(trans-4-stilbenyl)-4-methyl-morpholin-2-ol pH and temperature not specified in the publication 759144 2.5.1.21 0.0085 - 4-methyl-2-(4'-hydroxybiphenyl)-3,4-dihydro-2H-1,4-benzothiazin-2-ol pH and temperature not specified in the publication 759144 2.5.1.21 0.014 - 4-methyl-2-(4'-trifluromethyl-4-biphenyl)-3,4-dihydro-2H-1,4-benzothiazine-2-ol pH and temperature not specified in the publication 759144 2.5.1.21 0.0153 - [(1R,5R)-7-chloro-1-(2-methylpropyl)-2-oxo-5-phenyl-1,2,4,5-tetrahydro-3H-3-benzazepin-3-yl]acetic acid pH and temperature not specified in the publication 721801 2.5.1.21 0.0176 - carnosol pH 7.4, 37°C 759842 2.5.1.21 0.0184 - 11,12-di-O-methylcarnosol pH 7.4, 37°C 759842 2.5.1.21 0.02 - 1-[[(1S,5S)-7-chloro-5-(2,3-dimethoxyphenyl)-1-(2-methylpropyl)-2-oxo-1,2,4,5-tetrahydro-3H-3-benzazepin-3-yl]acetyl]piperidine-4-carboxylic acid pH and temperature not specified in the publication 721801 2.5.1.21 0.02 - ethyl [(1R,5S)-7-chloro-5-(2-chlorophenyl)-1-(2-methylpropyl)-2-oxo-1,2,4,5-tetrahydro-3H-3-benzazepin-3-yl]acetate pH and temperature not specified in the publication 721801 2.5.1.21 0.02 - [(1R,5S)-1-benzyl-7-chloro-5-(2-chlorophenyl)-2-oxo-1,2,4,5-tetrahydro-3H-3-benzazepin-3-yl]acetic acid pH and temperature not specified in the publication 721801 2.5.1.21 0.02 - [(1R,5S)-5-(2-chlorophenyl)-1-(2-methylpropyl)-2-oxo-1,2,4,5-tetrahydro-3H-3-benzazepin-3-yl]acetic acid pH and temperature not specified in the publication 721801 2.5.1.21 0.02 - [(1R,5S)-5-(2-chlorophenyl)-7-fluoro-1-(2-methylpropyl)-2-oxo-1,2,4,5-tetrahydro-3H-3-benzazepin-3-yl]acetic acid pH and temperature not specified in the publication 721801 2.5.1.21 0.02 - [(1R,5S)-5-(2-chlorophenyl)-7-methyl-1-(2-methylpropyl)-2-oxo-1,2,4,5-tetrahydro-3H-3-benzazepin-3-yl]acetic acid pH and temperature not specified in the publication 721801 2.5.1.21 0.02 - [(1R,5S)-7-chloro-5-(2-chlorophenyl)-1-(2-hydroxy-2-methylpropyl)-2-oxo-1,2,4,5-tetrahydro-3H-3-benzazepin-3-yl]acetic acid pH and temperature not specified in the publication 721801 2.5.1.21 0.0269 - rosmaquinone pH 7.4, 37°C 759842 2.5.1.21 0.028 - 4-methyl-2-phenyl-3,4-dihydro-2H-benzothiazin-2-ol pH and temperature not specified in the publication 759144 2.5.1.21 0.042 - 3-(trans-4-stilbenyl)octahydropyridino[2,1-c][1,4]oxazin-3-ol pH and temperature not specified in the publication 759144 2.5.1.21 0.05 - 4-methyl-2-phenyl-3,4-dihydro-2H-benzoxazin-2-ol pH and temperature not specified in the publication 759144 2.5.1.21 0.064 - CLSPHSMFC pH and temperature not specified in the publication 737480 2.5.1.21 0.0692 - galdosol pH 7.4, 37°C 759842 2.5.1.21 0.076 - SMFC pH and temperature not specified in the publication 737480 2.5.1.21 0.0802 - rosmanol pH 7.4, 37°C 759842 2.5.1.21 0.087 - CKTE pH and temperature not specified in the publication 737480 2.5.1.21 0.09 - WHQW pH and temperature not specified in the publication 737480 2.5.1.21 0.0903 - isorosmanol pH 7.4, 37°C 759842 2.5.1.21 0.0969 - rosmadial pH 7.4, 37°C 759842 2.5.1.21 0.378 - 11,12-diacetyl-carnosol pH 7.4, 37°C 759842 2.5.1.21 0.543 - 7alpha-methoxyrosmanol pH 7.4, 37°C 759842 2.5.1.21 1.336 - 7alpha-ethoxyrosmanol pH 7.4, 37°C 759842 2.5.1.21 1.524 - carnosol quinone pH 7.4, 37°C 759842