EC Number | Crystallization (Comment) | Organism |
---|---|---|
2.7.11.16 | in complex with CCG215022, hanging drop vapor diffusion method, using 100 mM HEPES, pH 7.5, 4% (v/v) ethylene glycol, and 12% (w/v) PEG3350 | Bos taurus |
EC Number | Inhibitors | Comment | Organism | Structure |
---|---|---|---|---|
2.7.11.16 | balanol | - |
Bos taurus | |
2.7.11.16 | CCG215022 | - |
Bos taurus | |
2.7.11.16 | GSK180736A | - |
Bos taurus | |
2.7.11.16 | paroxetine | - |
Bos taurus | |
2.7.11.16 | Takeda103A | - |
Bos taurus |
EC Number | Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|---|
2.7.11.16 | nucleus | - |
Bos taurus | 5634 | - |
EC Number | Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|---|
2.7.11.16 | ATP + [G-protein-coupled receptor] | Bos taurus | - |
ADP + [G-protein-coupled receptor]phosphate | - |
? |
EC Number | Organism | UniProt | Comment | Textmining |
---|---|---|---|---|
2.7.11.16 | Bos taurus | P43249 | - |
- |
EC Number | Purification (Comment) | Organism |
---|---|---|
2.7.11.16 | Ni-NTA column chromatography and S200 gel filtration | Bos taurus |
EC Number | Source Tissue | Comment | Organism | Textmining |
---|---|---|---|---|
2.7.11.16 | cardiomyocyte | - |
Bos taurus | - |
EC Number | Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|---|
2.7.11.16 | ATP + [G-protein-coupled receptor] | - |
Bos taurus | ADP + [G-protein-coupled receptor]phosphate | - |
? |
EC Number | Synonyms | Comment | Organism |
---|---|---|---|
2.7.11.16 | G protein-coupled receptor kinase 5 | - |
Bos taurus |
2.7.11.16 | GRK5 | - |
Bos taurus |