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Literature summary extracted from

  • Al-Aboudi, A.; Odeh, H.; Khalid, A.; Naz, Q.; Choudhary, M.I.
    Butyrylcholinesterase inhibitory activity of testosterone and some of its metabolites (2008), J. Enzyme Inhib. Med. Chem., 24, 553-558.
    View publication on PubMed

Inhibitors

EC Number Inhibitors Comment Organism Structure
3.1.1.8 1-dehydrotestosterone
-
 Equus caballus
3.1.1.8 11alpha,17beta-dihydroxyandrost-1,4-dien-3-one
-
 Equus caballus
3.1.1.8 11alpha-hydroxyandrost-1,4-dien-3,17-dione
-
 Equus caballus
3.1.1.8 11alpha-hydroxyandrost-4-en-3,17-dione
-
 Equus caballus
3.1.1.8 11alpha-hydroxytestolactone
-
 Equus caballus
3.1.1.8 11alpha-hydroxytestosterone
-
 Equus caballus
3.1.1.8 17beta-hydroxy-5alpha-androstan-3,6-dione
-
 Equus caballus
3.1.1.8 androst-1,4-dien-3,17-dione
-
 Equus caballus
3.1.1.8 androst-4-en-3,7-dione
-
 Equus caballus
3.1.1.8 galanthamine
-
 Equus caballus
3.1.1.8 additional information molecular docking analysis of inhibitors, overview Equus caballus
3.1.1.8 testolactone
-
 Equus caballus
3.1.1.8 testosterone
-
 Equus caballus

Localization

EC Number Localization Comment Organism GeneOntology No. Textmining
3.1.1.8 extracellular
-
 Equus caballus
-
-

Organism

EC Number Organism UniProt Comment Textmining
3.1.1.8 Equus caballus
-
-
-

Source Tissue

EC Number Source Tissue Comment Organism Textmining
3.1.1.8 serum
-
 Equus caballus
-

Synonyms

EC Number Synonyms Comment Organism
3.1.1.8 BChE
-
 Equus caballus
3.1.1.8 butyrylcholinesterase
-
 Equus caballus

Ki Value [mM]

EC Number Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
3.1.1.8 additional information
-
 additional information inhibition kinetics Equus caballus

IC50 Value

EC Number IC50 Value IC50 Value Maximum Comment Organism Inhibitor Structure
3.1.1.8 0.00155
-
-
 Equus caballus androst-4-en-3,7-dione
3.1.1.8 0.0085
-
-
 Equus caballus galanthamine
3.1.1.8 0.0209
-
-
 Equus caballus 1-dehydrotestosterone
3.1.1.8 0.0535
-
-
 Equus caballus testosterone
3.1.1.8 0.0615
-
-
 Equus caballus 11alpha,17beta-dihydroxyandrost-1,4-dien-3-one
3.1.1.8 0.089
-
-
 Equus caballus 11alpha-hydroxytestosterone
3.1.1.8 0.0959
-
-
 Equus caballus 17beta-hydroxy-5alpha-androstan-3,6-dione
3.1.1.8 0.1027
-
-
 Equus caballus androst-1,4-dien-3,17-dione
3.1.1.8 0.1413
-
-
 Equus caballus 11alpha-hydroxyandrost-4-en-3,17-dione
3.1.1.8 0.1425
-
-
 Equus caballus testolactone
3.1.1.8 0.1647
-
-
 Equus caballus 11alpha-hydroxyandrost-1,4-dien-3,17-dione
3.1.1.8 0.284
-
-
 Equus caballus 11alpha-hydroxytestolactone