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Literature summary extracted from

  • Wentland, M.P.; Raza, S.; Gao, Y.
    96-well plate colorimetric assay for Ki determination of (+-)-2-benzylsuccinic acid, an inhibitor of carboxypeptidase A: a laboratory experiment in drug discovery (2004), J. Chem. Educ., 81, 398-400.
No PubMed abstract available

Inhibitors

EC Number Inhibitors Comment Organism Structure
3.4.17.1 (+-)-2-benzylsuccinic acid
-
 Mammalia

KM Value [mM]

EC Number KM Value [mM] KM Value Maximum [mM] Substrate Comment Organism Structure
3.4.17.1 0.22
-
 Ac-Phe-ThiaPhe
-
 Mammalia

Metals/Ions

EC Number Metals/Ions Comment Organism Structure
3.4.17.1 Zn2+ zinc-metallopeptidase Mammalia

Organism

EC Number Organism UniProt Comment Textmining
3.4.17.1 Mammalia
-
-
-

Source Tissue

EC Number Source Tissue Comment Organism Textmining
3.4.17.1 pancreas
-
 Mammalia
-

Substrates and Products (Substrate)

EC Number Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
3.4.17.1 Ac-Phe-ThiaPhe + H2O
-
 Mammalia Phe + ThiaPhe
-
 ?
3.4.17.1 additional information the enzyme cleaves dipeptides or single amino acids from the C-terminus of polypeptides Mammalia ?
-
 ?

Synonyms

EC Number Synonyms Comment Organism
3.4.17.1 CPA
-
 Mammalia

Ki Value [mM]

EC Number Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
3.4.17.1 0.0011
-
 (+-)-2-benzylsuccinic acid
-
 Mammalia