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Literature summary extracted from

  • Burlando, B.; Magnelli, V.; Panfoli, I.; Berti, E.; Viarengo, A.
    Ligand-independent tyrosine kinase signalling in RTH 149 trout hepatoma cells: comparison among heavy metals and pro-oxidants (2003), Cell. Physiol. Biochem., 13, 147-154.
    View publication on PubMed

Activating Compound

EC Number Activating Compound Comment Organism Structure
2.7.10.2 H2O2 increases tyrosine phosphorylation in vivo, genistein decreases the activating effect Oncorhynchus mykiss

Inhibitors

EC Number Inhibitors Comment Organism Structure
2.7.10.2 genistein
-
Oncorhynchus mykiss

Metals/Ions

EC Number Metals/Ions Comment Organism Structure
2.7.10.2 Cu2+ increases tyrosine phosphorylation in vivo, prevented by preincubation with genistein Oncorhynchus mykiss
2.7.10.2 Hg2+ increases tyrosine phosphorylation in vivo, genistein decreases the activating effect Oncorhynchus mykiss

Natural Substrates/ Products (Substrates)

EC Number Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
2.7.10.2 ATP + a [protein]-L-tyrosine Oncorhynchus mykiss
-
ADP + a [protein]-L-tyrosine phosphate
-
?
2.7.10.2 additional information Oncorhynchus mykiss enzyme is involved in cell growth, differentiation, and apoptosis ?
-
?

Organism

EC Number Organism UniProt Comment Textmining
2.7.10.2 Oncorhynchus mykiss
-
-
-

Source Tissue

EC Number Source Tissue Comment Organism Textmining
2.7.10.2 hepatoma cell
-
Oncorhynchus mykiss
-
2.7.10.2 RTH-149 cell hepatoma cell line Oncorhynchus mykiss
-

Substrates and Products (Substrate)

EC Number Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
2.7.10.2 ATP + a [protein]-L-tyrosine
-
Oncorhynchus mykiss ADP + a [protein]-L-tyrosine phosphate
-
?
2.7.10.2 additional information enzyme is involved in cell growth, differentiation, and apoptosis Oncorhynchus mykiss ?
-
?

Synonyms

EC Number Synonyms Comment Organism
2.7.10.2 non-receptor tyrosine kinase
-
Oncorhynchus mykiss