EC Number | Activating Compound | Comment | Organism | Structure |
---|---|---|---|---|
3.4.22.15 | Cys | activates | Rattus norvegicus | |
3.4.22.15 | Cys | activates | Cyprinus carpio |
EC Number | Inhibitors | Comment | Organism | Structure |
---|---|---|---|---|
3.4.22.15 | 1,10-phenanthroline | - |
Cyprinus carpio | |
3.4.22.15 | 5,5'-dithiobis(2-nitrobenzoic acid) | - |
Cyprinus carpio | |
3.4.22.15 | 5,5'-dithiobis(2-nitrobenzoic acid) | - |
Rattus norvegicus | |
3.4.22.15 | AgNO3 | - |
Cyprinus carpio | |
3.4.22.15 | antipain | - |
Cyprinus carpio | |
3.4.22.15 | CdCl2 | - |
Cyprinus carpio | |
3.4.22.15 | chymostatin | - |
Cyprinus carpio | |
3.4.22.15 | CoCl2 | partial | Cyprinus carpio | |
3.4.22.15 | CuCl2 | - |
Cyprinus carpio | |
3.4.22.15 | FeCl3 | - |
Cyprinus carpio | |
3.4.22.15 | Hg2+ | HgCl2 | Cyprinus carpio | |
3.4.22.15 | Hg2+ | - |
Rattus norvegicus | |
3.4.22.15 | leupeptin | - |
Cyprinus carpio | |
3.4.22.15 | leupeptin | - |
Rattus norvegicus | |
3.4.22.15 | PCMB | - |
Cyprinus carpio | |
3.4.22.15 | PCMB | - |
Rattus norvegicus | |
3.4.22.15 | SnCl2 < | partial | Cyprinus carpio | |
3.4.22.15 | trans-epoxysuccinyl-L-leucylamido-(4-guanidino)butane | - |
Cyprinus carpio | |
3.4.22.15 | trans-epoxysuccinyl-L-leucylamido-(4-guanidino)butane | i.e. E-64, in vivo, the inhibitor is transported to the liver cytosol in the free form in the blood and permeated into the lysosomes, where it binds to, and inactivates the enzyme | Rattus norvegicus | |
3.4.22.15 | Zn(CH3COO)2 | - |
Cyprinus carpio |
EC Number | KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|---|
3.4.22.15 | 0.03416 | - |
benzyloxycarbonyl-Phe-Arg-4-methylcoumarin 7-amide | - |
Cyprinus carpio | |
3.4.22.15 | 0.04371 | - |
Pro-Phe-Arg-4-methylcoumarin 7-amide | - |
Cyprinus carpio | |
3.4.22.15 | 0.1417 | - |
tert-butyloxycarbonyl-Val-Leu-Lys-4-methylcoumarin 7-amide | - |
Cyprinus carpio |
EC Number | Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|---|
3.4.22.15 | lysosome | - |
Rattus norvegicus | 5764 | - |
EC Number | Molecular Weight [Da] | Molecular Weight Maximum [Da] | Comment | Organism |
---|---|---|---|---|
3.4.22.15 | 24000 | - |
x * 24000 + x * 30000, SDS-PAGE under reducing conditions | Cyprinus carpio |
3.4.22.15 | 30000 | - |
gel filtration | Cyprinus carpio |
EC Number | Organism | UniProt | Comment | Textmining |
---|---|---|---|---|
3.4.22.15 | Cyprinus carpio | - |
- |
- |
3.4.22.15 | Rattus norvegicus | - |
- |
- |
EC Number | Purification (Comment) | Organism |
---|---|---|
3.4.22.15 | - |
Cyprinus carpio |
EC Number | Source Tissue | Comment | Organism | Textmining |
---|---|---|---|---|
3.4.22.15 | hepatopancreas | - |
Cyprinus carpio | - |
3.4.22.15 | liver | - |
Rattus norvegicus | - |
EC Number | Specific Activity Minimum [µmol/min/mg] | Specific Activity Maximum [µmol/min/mg] | Comment | Organism |
---|---|---|---|---|
3.4.22.15 | additional information | - |
- |
Cyprinus carpio |
EC Number | Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|---|
3.4.22.15 | benzyloxycarbonyl-Phe-Arg-4-methylcoumarin 7-amide + H2O | - |
Rattus norvegicus | ? | - |
? | |
3.4.22.15 | benzyloxycarbonyl-Phe-Arg-4-methylcoumarin 7-amide + H2O | - |
Cyprinus carpio | ? | - |
? | |
3.4.22.15 | Pro-Phe-Arg-4-methylcoumarin 7-amide + H2O | - |
Cyprinus carpio | ? | - |
? | |
3.4.22.15 | tert-butyloxycarbonyl-Val-Leu-Lys-4-methylcoumarin 7-amide + H2O | - |
Cyprinus carpio | ? | - |
? |
EC Number | Subunits | Comment | Organism |
---|---|---|---|
3.4.22.15 | ? | - |
Rattus norvegicus |
3.4.22.15 | ? | x * 24000 + x * 30000, SDS-PAGE under reducing conditions | Cyprinus carpio |
EC Number | Temperature Optimum [°C] | Temperature Optimum Maximum [°C] | Comment | Organism |
---|---|---|---|---|
3.4.22.15 | 50 | - |
hydrolysis of benzyloxycarbonyl-Phe-Arg-4-methylcoumarin 7-amide | Cyprinus carpio |
EC Number | Temperature Minimum [°C] | Temperature Maximum [°C] | Comment | Organism |
---|---|---|---|---|
3.4.22.15 | 30 | - |
less than half maximal activity below 30°C and above 60°C | Cyprinus carpio |
EC Number | Temperature Stability Minimum [°C] | Temperature Stability Maximum [°C] | Comment | Organism |
---|---|---|---|---|
3.4.22.15 | 40 | - |
stable below | Cyprinus carpio |
EC Number | Turnover Number Minimum [1/s] | Turnover Number Maximum [1/s] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|---|
3.4.22.15 | 1.52 | - |
Pro-Phe-Arg-4-methylcoumarin 7-amide | - |
Cyprinus carpio | |
3.4.22.15 | 1.67 | - |
tert-butyloxycarbonyl-Val-Leu-Lys-4-methylcoumarin 7-amide | - |
Cyprinus carpio | |
3.4.22.15 | 9.5 | - |
benzyloxycarbonyl-Phe-Arg-4-methylcoumarin 7-amide | - |
Cyprinus carpio |
EC Number | pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|---|
3.4.22.15 | 5.5 | 6 | hydrolysis of benzyloxycarbonyl-Phe-Arg-4-methylcoumarin 7-amide | Cyprinus carpio |
EC Number | pH Stability | pH Stability Maximum | Comment | Organism |
---|---|---|---|---|
3.4.22.15 | 5 | 6.5 | stable | Cyprinus carpio |