EC Number | Inhibitors | Comment | Organism | Structure |
---|---|---|---|---|
2.8.3.5 | 2,2-Difluorosuccinate | strong | Rattus norvegicus | |
2.8.3.5 | 3-Sulfopropanoate | - |
Rattus norvegicus | |
2.8.3.5 | acetoacetate | - |
Rattus norvegicus | |
2.8.3.5 | acetylene dicarboxylate | weak | Rattus norvegicus | |
2.8.3.5 | Maleamate | reversible, competitive | Rattus norvegicus | |
2.8.3.5 | Maleimide | succinate or acetoacetate protects | Rattus norvegicus | |
2.8.3.5 | malonate | kinetics | Rattus norvegicus | |
2.8.3.5 | Monomethylsuccinate | competitive | Rattus norvegicus | |
2.8.3.5 | additional information | no inhibition by glutarate, adipate, cis- or trans-cyclobutane-1,2-dicarboxylate, cis- or trans-cyclohexane-1,2-dicarboxylate, methylsuccinate, mercaptosuccinate, malate, aspartate, succinimide or iodoacetamide | Rattus norvegicus | |
2.8.3.5 | N-ethylmaleamate | reversible, competitive | Rattus norvegicus | |
2.8.3.5 | N-ethylmaleimide | succinate or acetoacetate protects | Rattus norvegicus | |
2.8.3.5 | oxalate | kinetics | Rattus norvegicus | |
2.8.3.5 | Perfluorosuccinate | strong | Rattus norvegicus | |
2.8.3.5 | succinamate | competitive | Rattus norvegicus | |
2.8.3.5 | succinate | product inhibition | Rattus norvegicus |
EC Number | KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|---|
2.8.3.5 | 0.04 | - |
acetoacetyl-CoA | pH 8.1, 25°C | Rattus norvegicus | |
2.8.3.5 | 0.28 | - |
succinyl-CoA | pH 8.1, 25°C | Rattus norvegicus | |
2.8.3.5 | 0.44 | - |
acetoacetate | pH 8.1, 25°C | Rattus norvegicus | |
2.8.3.5 | 28 | - |
succinate | cosusbstrate: acetoacetyl-CoA, pH 8.1, 25°C | Rattus norvegicus | |
2.8.3.5 | 35 | - |
Maleate | cosusbstrate: acetoacetyl-CoA, pH 8.1, 25°C | Rattus norvegicus |
EC Number | Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|---|
2.8.3.5 | mitochondrion | - |
Rattus norvegicus | 5739 | - |
EC Number | Organism | UniProt | Comment | Textmining |
---|---|---|---|---|
2.8.3.5 | Rattus norvegicus | - |
male adult Buffalo | - |
EC Number | Purification (Comment) | Organism |
---|---|---|
2.8.3.5 | partial | Rattus norvegicus |
EC Number | Source Tissue | Comment | Organism | Textmining |
---|---|---|---|---|
2.8.3.5 | heart | - |
Rattus norvegicus | - |
EC Number | Specific Activity Minimum [µmol/min/mg] | Specific Activity Maximum [µmol/min/mg] | Comment | Organism |
---|---|---|---|---|
2.8.3.5 | 2.88 | - |
- |
Rattus norvegicus |
EC Number | Storage Stability | Organism |
---|---|---|
2.8.3.5 | frozen, partially purified preparation in phosphate solution, less than 10% loss of activity within 1-2 weeks | Rattus norvegicus |
EC Number | Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|---|
2.8.3.5 | additional information | no substrates are diacids with connecting chain lengths of 3 or more methylene groups | Rattus norvegicus | ? | - |
? | |
2.8.3.5 | succinyl-CoA + acetoacetate | - |
Rattus norvegicus | succinate + acetoacetyl-CoA | - |
r | |
2.8.3.5 | succinyl-CoA + maleate | - |
Rattus norvegicus | succinate + maleyl-CoA | - |
? |
EC Number | Temperature Optimum [°C] | Temperature Optimum Maximum [°C] | Comment | Organism |
---|---|---|---|---|
2.8.3.5 | 25 | - |
assay at | Rattus norvegicus |
EC Number | Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|---|
2.8.3.5 | 0.72 | - |
succinate | pH 8.1, 25°C | Rattus norvegicus | |
2.8.3.5 | 3.7 | - |
acetoacetate | pH 8.1, 25°C | Rattus norvegicus | |
2.8.3.5 | 6.4 | - |
2,2-Difluorosuccinate | pH 8.1, 25°C | Rattus norvegicus | |
2.8.3.5 | 15 | - |
oxalate | pH 8.1, 25°C | Rattus norvegicus | |
2.8.3.5 | 18 | - |
Perfluorosuccinate | pH 8.1, 25°C | Rattus norvegicus | |
2.8.3.5 | 21 | - |
malonate | pH 8.1, 25°C | Rattus norvegicus |