EC Number | Inhibitors | Comment | Organism | Structure |
---|---|---|---|---|
2.4.2.30 | 1-methylnicotinamide chloride | IC50: 1.7 mM | Bos taurus | |
2.4.2.30 | 2-Aminobenzamide | IC50: 0.1 mM | Bos taurus | |
2.4.2.30 | 3-aminobenzamide | IC50: 0.0054 | Bos taurus | |
2.4.2.30 | 3-isobutyl-1-methylxanthine | IC50: 3.1 mM | Bos taurus | |
2.4.2.30 | 3-Methoxybenzamide | IC50: 0.0034 mM | Bos taurus | |
2.4.2.30 | 4-Aminobenzamide | IC50: 0.4 mM | Bos taurus | |
2.4.2.30 | 5-bromodeoxyuridine | IC50: 0.015 mM | Bos taurus | |
2.4.2.30 | 5-Methylnicotinamide | IC50: 0.07 | Bos taurus | |
2.4.2.30 | 8-Methylnicotinamide | IC50: 7.8 mM | Bos taurus | |
2.4.2.30 | Benzamide | IC50: 0.0033 mM | Bos taurus | |
2.4.2.30 | Caffeine | IC50: 1.4 mM | Bos taurus | |
2.4.2.30 | hypoxanthine | IC50: 1.7 mM | Bos taurus | |
2.4.2.30 | Isonicotinate hydrazide | IC50: 4.8 MM | Bos taurus | |
2.4.2.30 | nicotinamide | IC50: 0.031 mM | Bos taurus | |
2.4.2.30 | Pyrazinamide | IC50: 0.13 mM | Bos taurus | |
2.4.2.30 | Theobromine | IC50: 0.11 mM | Bos taurus | |
2.4.2.30 | theophylline | IC50: 0.0046 | Bos taurus | |
2.4.2.30 | thymidine | IC50: 0.043 | Bos taurus | |
2.4.2.30 | Zn2+ | ZnCl2, IC50: 0.077 mM | Bos taurus |
EC Number | Organism | UniProt | Comment | Textmining |
---|---|---|---|---|
2.4.2.30 | Bos taurus | - |
calf | - |
EC Number | Source Tissue | Comment | Organism | Textmining |
---|---|---|---|---|
2.4.2.30 | thymus | - |
Bos taurus | - |
EC Number | Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|---|
2.4.2.30 | NAD+ + (ADP-D-ribosyl)n-acceptor | - |
Bos taurus | nicotinamide + (ADP-D-ribosyl)n+1-acceptor | - |
? |
EC Number | IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|---|
2.4.2.30 | 0.0033 | - |
IC50: 0.0033 mM | Bos taurus | Benzamide | |
2.4.2.30 | 0.0034 | - |
IC50: 0.0034 mM | Bos taurus | 3-Methoxybenzamide | |
2.4.2.30 | 0.0054 | - |
IC50: 0.0054 | Bos taurus | 3-aminobenzamide | |
2.4.2.30 | 0.015 | - |
IC50: 0.015 mM | Bos taurus | 5-bromodeoxyuridine | |
2.4.2.30 | 0.031 | - |
IC50: 0.031 mM | Bos taurus | nicotinamide | |
2.4.2.30 | 0.043 | - |
IC50: 0.043 mM | Bos taurus | thymidine | |
2.4.2.30 | 0.046 | - |
IC50: 0.046 mM | Bos taurus | theophylline | |
2.4.2.30 | 0.07 | - |
IC50: 0.07 mM | Bos taurus | 5-Methylnicotinamide | |
2.4.2.30 | 0.077 | - |
ZnCl2, IC50: 0.077 mM | Bos taurus | Zn2+ | |
2.4.2.30 | 0.1 | - |
IC50: 0.1 mM | Bos taurus | 2-Aminobenzamide | |
2.4.2.30 | 0.11 | - |
IC50: 0.11 mM | Bos taurus | Theobromine | |
2.4.2.30 | 0.13 | - |
IC50: 0.13 mM | Bos taurus | Pyrazinamide | |
2.4.2.30 | 0.4 | - |
IC50: 0.4 mM | Bos taurus | 4-Aminobenzamide | |
2.4.2.30 | 1.4 | - |
IC50: 1.4 mM | Bos taurus | Caffeine | |
2.4.2.30 | 1.7 | - |
IC50: 1.7 mM | Bos taurus | hypoxanthine | |
2.4.2.30 | 1.7 | - |
IC50: 1.7 mM | Bos taurus | 1-methylnicotinamide chloride | |
2.4.2.30 | 3.1 | - |
IC50: 3.1 mM | Bos taurus | 3-isobutyl-1-methylxanthine | |
2.4.2.30 | 4.8 | - |
IC50: 4.8 mM | Bos taurus | Isonicotinate hydrazide | |
2.4.2.30 | 7.8 | - |
IC50: 7.8 mM | Bos taurus | 8-Methylnicotinamide |