EC Number | Inhibitors | Comment | Organism | Structure |
---|---|---|---|---|
3.4.17.21 | 1,10-phenanthroline | 1 mM, 90% inhibition | Rattus norvegicus | |
3.4.17.21 | 2-oxoglutarate | 0.1 mM, 46% inhibition | Rattus norvegicus | |
3.4.17.21 | Ala-Glu | 0.0061 mM, 50% inhibition | Rattus norvegicus | |
3.4.17.21 | Asp-Ala | 0.1 mM, 26% inhibition | Rattus norvegicus | |
3.4.17.21 | Asp-Asp | 0.1 mM, 42% inhibition | Rattus norvegicus | |
3.4.17.21 | Asp-Glu | 0.0024 mM, 50% inhibition | Rattus norvegicus | |
3.4.17.21 | Asp-Phe | 0.1 mM, 22% inhibition | Rattus norvegicus | |
3.4.17.21 | aspartate | 0.1 mM, 42% inhibition | Rattus norvegicus | |
3.4.17.21 | bestatin | 0.29 mM, 79% inhibition | Rattus norvegicus | |
3.4.17.21 | Cd2+ | - |
Rattus norvegicus | |
3.4.17.21 | Cu2+ | - |
Rattus norvegicus | |
3.4.17.21 | cysteate | 0.1 mM, 40% inhibition | Rattus norvegicus | |
3.4.17.21 | cysteine sulfinate | 0.1 mM, 42% inhibition | Rattus norvegicus | |
3.4.17.21 | D-Glu-D-Glu | 0.1 mM, 50% inhibition | Rattus norvegicus | |
3.4.17.21 | dithiothreitol | 1 mM, 94.8% inhibition | Rattus norvegicus | |
3.4.17.21 | EDTA | 1 mM, 96.3% inhibition | Rattus norvegicus | |
3.4.17.21 | EGTA | 1 mM, 92% inhibition | Rattus norvegicus | |
3.4.17.21 | Fe3+ | - |
Rattus norvegicus | |
3.4.17.21 | gamma-Glu-Glu | 0.0095 mM, 50% inhibition | Rattus norvegicus | |
3.4.17.21 | Glu-Asp | 0.1 mM, 27% inhibition | Rattus norvegicus | |
3.4.17.21 | Glu-Glu | 0.00075 mM, 50% inhibition | Rattus norvegicus | |
3.4.17.21 | Glu-Glu-Glu | 0.062 mM, 50% inhibition | Rattus norvegicus | |
3.4.17.21 | glutathione | i.e. gamma-Glu-Cys-Gly, 0.019 mM, 50% inhibition | Rattus norvegicus | |
3.4.17.21 | Gly-Glu | 0.008 mM, 50% inhibition | Rattus norvegicus | |
3.4.17.21 | Gly-Gly-Glu | 0.00098 mM, 50% inhibition | Rattus norvegicus | |
3.4.17.21 | Ibotenate | 0.1 mM, 45% inhibition | Rattus norvegicus | |
3.4.17.21 | iodoacetate | 1 mM, 38% inhibition | Rattus norvegicus | |
3.4.17.21 | L-2-Amino-4-phosphonobutanoate | 0.1 mM, 37% inhibition | Rattus norvegicus | |
3.4.17.21 | L-Glu | 0.032 mM, 50% inhibition | Rattus norvegicus | |
3.4.17.21 | additional information | not inhibitory are pepstatin, iodoacetamide, amastatin | Rattus norvegicus | |
3.4.17.21 | N-Acetyl-Asp-Gln | 0.1 mM, 49% inhibition | Rattus norvegicus | |
3.4.17.21 | N-Acetyl-Asp-Glu-Asp | 0.1 mM, 49% inhibition | Rattus norvegicus | |
3.4.17.21 | N-Acetyl-Asp-Ser-Gly | 0.1 mM, 37% inhibition | Rattus norvegicus | |
3.4.17.21 | N-Acetyl-Glu-Asp | 0.036 mM, 50% inhibition | Rattus norvegicus | |
3.4.17.21 | N-Acetyl-Glu-Glu | 0.00031 mM, 50% inhibition | Rattus norvegicus | |
3.4.17.21 | N-acetyl-L-Asp | 0.1 mM, 38% inhibition | Rattus norvegicus | |
3.4.17.21 | N-Acetyl-L-Asp-L-Glu | 0.00054 mM, 50% inhibition | Rattus norvegicus | |
3.4.17.21 | N-acetyl-L-Glu | 0.058 mM, 50% inhibition | Rattus norvegicus | |
3.4.17.21 | Phe-Glu | 0.077 mM, 50% inhibition | Rattus norvegicus | |
3.4.17.21 | PO43- | - |
Rattus norvegicus | |
3.4.17.21 | puromycin | 0.5 mM, 55% inhibition | Rattus norvegicus | |
3.4.17.21 | pyroglutamate | 0.1 mM, 27% inhibition | Rattus norvegicus | |
3.4.17.21 | quinolinate | 0.1 mM, 41% inhibition | Rattus norvegicus | |
3.4.17.21 | Quisqualic acid | 0.00048 mM, 50% inhibition | Rattus norvegicus | |
3.4.17.21 | Serine O-sulfate | 0.042 mM, 50% inhibition | Rattus norvegicus | |
3.4.17.21 | SO42- | - |
Rattus norvegicus | |
3.4.17.21 | Tyr-Glu | 0.1 mM, 45% inhibition | Rattus norvegicus | |
3.4.17.21 | Val-Glu-Glu | 0.036 mM, 50% inhibition | Rattus norvegicus | |
3.4.17.21 | Zn2+ | - |
Rattus norvegicus |
EC Number | KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|---|
3.4.17.21 | 540 | - |
N-Acetyl-L-Asp-L-Glu | - |
Rattus norvegicus |
EC Number | Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|---|
3.4.17.21 | membrane | - |
Rattus norvegicus | 16020 | - |
EC Number | Metals/Ions | Comment | Organism | Structure |
---|---|---|---|---|
3.4.17.21 | Br- | 2 mM, activation | Rattus norvegicus | |
3.4.17.21 | Ca2+ | activation | Rattus norvegicus | |
3.4.17.21 | Cl- | 2 mM, activation | Rattus norvegicus | |
3.4.17.21 | Co2+ | activation | Rattus norvegicus | |
3.4.17.21 | F- | 100 mM, 20% of the activity compared to Cl- | Rattus norvegicus | |
3.4.17.21 | I- | 2 mM, activation | Rattus norvegicus | |
3.4.17.21 | Mg2+ | activation | Rattus norvegicus | |
3.4.17.21 | Mn2+ | activation | Rattus norvegicus | |
3.4.17.21 | NO3- | 2 mM , activation | Rattus norvegicus | |
3.4.17.21 | Sr2+ | activation | Rattus norvegicus |
EC Number | Organism | UniProt | Comment | Textmining |
---|---|---|---|---|
3.4.17.21 | Rattus norvegicus | - |
- |
- |
EC Number | Source Tissue | Comment | Organism | Textmining |
---|---|---|---|---|
3.4.17.21 | brain | forebrain | Rattus norvegicus | - |
EC Number | Specific Activity Minimum [µmol/min/mg] | Specific Activity Maximum [µmol/min/mg] | Comment | Organism |
---|---|---|---|---|
3.4.17.21 | additional information | - |
assay method | Rattus norvegicus |
EC Number | Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|---|
3.4.17.21 | N-Acetyl-L-Asp-L-Glu + H2O | - |
Rattus norvegicus | N-Acetyl-L-Asp + L-Glu | - |
? |
EC Number | Temperature Optimum [°C] | Temperature Optimum Maximum [°C] | Comment | Organism |
---|---|---|---|---|
3.4.17.21 | 37 | - |
- |
Rattus norvegicus |
EC Number | Temperature Minimum [°C] | Temperature Maximum [°C] | Comment | Organism |
---|---|---|---|---|
3.4.17.21 | 25 | 80 | more than 50% of maximal activity in this range | Rattus norvegicus |
EC Number | pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|---|
3.4.17.21 | 7 | - |
- |
Rattus norvegicus |
EC Number | pH Minimum | pH Maximum | Comment | Organism |
---|---|---|---|---|
3.4.17.21 | 6 | 7.4 | more than 50% of maximal activity in this range | Rattus norvegicus |
EC Number | Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|---|
3.4.17.21 | 0.00031 | - |
N-Acetyl-Glu-Glu | - |
Rattus norvegicus | |
3.4.17.21 | 0.00054 | - |
N-Acetyl-L-Asp-L-Glu | - |
Rattus norvegicus | |
3.4.17.21 | 0.00075 | - |
Glu-Glu | - |
Rattus norvegicus | |
3.4.17.21 | 0.00098 | - |
Gly-Gly-Glu | - |
Rattus norvegicus | |
3.4.17.21 | 0.0024 | - |
Asp-Glu | - |
Rattus norvegicus | |
3.4.17.21 | 0.008 | - |
Gly-Glu | - |
Rattus norvegicus | |
3.4.17.21 | 0.019 | - |
glutathione | i.e. gamma-Glu-Cys-Gly | Rattus norvegicus | |
3.4.17.21 | 0.036 | - |
N-Acetyl-Glu-Asp | - |
Rattus norvegicus | |
3.4.17.21 | 0.036 | - |
Val-Glu-Glu | - |
Rattus norvegicus | |
3.4.17.21 | 0.042 | - |
Serine O-sulfate | - |
Rattus norvegicus | |
3.4.17.21 | 0.058 | - |
N-acetyl-L-Glu | - |
Rattus norvegicus | |
3.4.17.21 | 0.061 | - |
Ala-Glu | - |
Rattus norvegicus | |
3.4.17.21 | 0.062 | - |
Glu-Glu-Glu | - |
Rattus norvegicus | |
3.4.17.21 | 0.077 | - |
Phe-Glu | - |
Rattus norvegicus | |
3.4.17.21 | 0.095 | - |
gamma-Glu-Glu | - |
Rattus norvegicus | |
3.4.17.21 | 0.1 | - |
D-Glu-D-Glu | - |
Rattus norvegicus |