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Literature summary for 7.2.2.13 extracted from

  • Garcia, D.G.; Bianco, E.M.; Santos, M.D.; Pereira, R.C.; Faria, M.V.; Teixeira, V.L.; Burth, P.
    Inhibition of mammal Na(+)K(+)-ATPase by diterpenes extracted from the Brazilian brown alga Dictyota cervicornis (2009), Phytother. Res., 23, 943-947.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
4,7-diacetoxy-14-hydroxydolast-1(15),8-diene
-
Cavia porcellus
4-acetoxy-9,14-dihydroxydolast-1(15),7-diene
-
Cavia porcellus
oleic acid
-
Cavia porcellus
Ouabain
-
Cavia porcellus

Organism

Organism UniProt Comment Textmining
Cavia porcellus
-
-
-

Purification (Commentary)

Purification (Comment) Organism
-
Cavia porcellus

Source Tissue

Source Tissue Comment Organism Textmining
brain mainly alpha2- and alpha3 isoform Cavia porcellus
-
kidney alpha1-isoform Cavia porcellus
-

Synonyms

Synonyms Comment Organism
Na+-K+-ATPase
-
Cavia porcellus

IC50 Value

IC50 Value IC50 Value Maximum Comment Organism Inhibitor Structure
0.0016
-
enzym preparation from kidney Cavia porcellus Ouabain
0.115
-
enzym preparation from kidney Cavia porcellus oleic acid
0.171
-
enzym preparation from kidney Cavia porcellus 4,7-diacetoxy-14-hydroxydolast-1(15),8-diene