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Literature summary for 7.1.2.2 extracted from

  • Johnson, R.M.; Allen, C.; Melman, S.D.; Waller, A.; Young, S.M.; Sklar, L.A.; Parra, K.J.
    Identification of inhibitors of vacuolar proton-translocating ATPase pumps in yeast by high-throughput screening flow cytometry (2010), Anal. Biochem., 398, 203-211.
    View publication on PubMedView publication on EuropePMC

Application

Application Comment Organism
drug development the enzyme is a target for development of specific inhibitors Saccharomyces cerevisiae

Inhibitors

Inhibitors Comment Organism Structure
concanamycin A
-
Saccharomyces cerevisiae
Disulfiram
-
Saccharomyces cerevisiae
additional information inhibitor screening, overview Saccharomyces cerevisiae

Localization

Localization Comment Organism GeneOntology No. Textmining
additional information enzyme localization study, overview Saccharomyces cerevisiae
-
-
vacuolar membrane
-
Saccharomyces cerevisiae 5774
-

Metals/Ions

Metals/Ions Comment Organism Structure
Mg2+ required Saccharomyces cerevisiae

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
ATP + H2O + H+/in Saccharomyces cerevisiae
-
ADP + phosphate + H+/out
-
?
ATP + H2O + H+/in Saccharomyces cerevisiae BY4741
-
ADP + phosphate + H+/out
-
?

Organism

Organism UniProt Comment Textmining
Saccharomyces cerevisiae
-
-
-
Saccharomyces cerevisiae BY4741
-
-
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
ATP + H2O + H+/in
-
Saccharomyces cerevisiae ADP + phosphate + H+/out
-
?
ATP + H2O + H+/in
-
Saccharomyces cerevisiae BY4741 ADP + phosphate + H+/out
-
?

Synonyms

Synonyms Comment Organism
V-ATPase
-
Saccharomyces cerevisiae
vacuolar proton-translocating ATPase
-
Saccharomyces cerevisiae

pH Optimum

pH Optimum Minimum pH Optimum Maximum Comment Organism
6.9 7 assay at Saccharomyces cerevisiae