Crystallization (Comment) | Organism |
---|---|
hanging drop method, GDP-2'-deoxy-6-phosphoryl-IMP complex | Mus musculus |
hanging drop method, GDP-2'-deoxy-6-phosphoryl-IMP-hadacidin complex | Escherichia coli |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
Hadacidin | - |
Escherichia coli | |
Hadacidin | - |
Mus musculus |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.004 | - |
L-Asp | 22°C, cosubstrate: 2'-dIMP | Mus musculus | |
0.013 | - |
L-Asp | 22°C, cosubstrate: 2'-dIMP | Escherichia coli | |
0.015 | - |
GTP | 22°C, cosubstrate: 2'-dIMP | Mus musculus | |
0.021 | - |
GTP | 22°C, cosubstrate: 2'-dIMP | Escherichia coli | |
0.026 | - |
GTP | 22°C, cosubstrate: IMP | Escherichia coli | |
0.028 | - |
IMP | 22°C | Escherichia coli | |
0.041 | - |
2'-dIMP | 22°C | Escherichia coli | |
0.058 | - |
2'-dIMP | 22°C | Mus musculus | |
0.23 | - |
L-Asp | 22°C, cosubstrate: dIMP | Escherichia coli |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Escherichia coli | P0A7D4 | - |
- |
Mus musculus | P28650 | - |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
muscle | - |
Mus musculus | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + IMP + L-Asp | - |
Escherichia coli | GDP + phosphate + adenylosuccinate | - |
? | |
ATP + IMP + L-Asp | - |
Mus musculus | GDP + phosphate + adenylosuccinate | - |
? | |
GTP + 2'-dIMP + L-Asp | - |
Escherichia coli | GDP + phosphate + 2'-deoxysuccinoAMP | - |
? | |
GTP + 2'-dIMP + L-Asp | - |
Mus musculus | GDP + phosphate + 2'-deoxysuccinoAMP | - |
? |
Turnover Number Minimum [1/s] | Turnover Number Maximum [1/s] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.96 | - |
2'-dIMP | 22°C | Escherichia coli | |
0.96 | - |
GTP | 22°C, cosubstrate: 2'-dIMP | Escherichia coli | |
0.96 | - |
L-Asp | 22°C, cosubstrate: 2'-dIMP | Escherichia coli | |
1 | - |
IMP | 22°C | Escherichia coli | |
1 | - |
GTP | 22°C, cosubstrate: IMP | Escherichia coli | |
1 | - |
L-Asp | 22°C, cosubstrate: IMP | Escherichia coli | |
5.5 | - |
2'-dIMP | 22°C | Mus musculus | |
5.5 | - |
GTP | 22°C, cosubstrate: 2'-dIMP | Mus musculus | |
5.5 | - |
L-Asp | 22°C, cosubstrate: 2'-dIMP | Mus musculus |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.00032 | - |
Hadacidin | reaction with IMP | Mus musculus | |
0.00049 | - |
Hadacidin | 22°C, reaction with IMP | Escherichia coli | |
0.014 | - |
Hadacidin | reaction with 2'-dIMP | Mus musculus | |
0.017 | - |
Hadacidin | 22°C, reaction with 2'-dIMP | Escherichia coli |