Inhibitors | Comment | Organism | Structure |
---|---|---|---|
(2'R,6'S)-9-[6'-([[N-(D-biotinoyl)sulfamoyl]oxy]methyl)morpholin-2'-yl]adenine | nucleoside-based inhibitor, KD value 0.324 nM | Mycobacterium tuberculosis | |
2'-amino-5'-[N-(D-biotinoyl)sulfamoyl]amino-3',5'-dideoxyadenosine | nucleoside-based inhibitor, KD value 0.627 nM | Mycobacterium tuberculosis | |
9-[2'-azido-5'-O-[N-(D-biotinoyl)sulfamoyl]-2'-deoxy-beta-D-arabinofuranosyl]adenine | nucleoside-based inhibitor, KD value 0.027 nM. Strongest binding inhibitor in series | Mycobacterium tuberculosis |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Mycobacterium tuberculosis | I6YFP0 | - |
- |
Mycobacterium tuberculosis H37Rv | I6YFP0 | - |
- |