Cloned (Comment) | Organism |
---|---|
expression in Sf9 cells | Mus musculus |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
CTP | - |
Mus musculus | |
cytidine 5'-(gamma-thio)triphosphate | - |
Mus musculus | |
GTP | - |
Mus musculus | |
guanosine 5'-(beta,gamma-imido)triphosphate | - |
Mus musculus | |
guanosine 5'-(gamma-thio)triphosphate | - |
Mus musculus | |
inosine 5'-(beta,gamma-imido)triphosphate | - |
Mus musculus | |
inosine 5'-(gamma-thio)triphosphate | - |
Mus musculus | |
ITP | - |
Mus musculus | |
additional information | inhibition studies of the purified catalytic subunits in the presence of forskolin | Mus musculus | |
uridine 5'-(beta,gamma-imido)triphosphate | - |
Mus musculus | |
uridine 5'-(gamma-thio)triphosphate | - |
Mus musculus | |
UTP | - |
Mus musculus | |
xanthosine 5'-(beta,gamma-imido)triphosphate | - |
Mus musculus | |
xanthosine 5'-(gamma-thio)triphosphate | - |
Mus musculus | |
XTP | - |
Mus musculus |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.1 | - |
ATP | Sf9, Mn2+, pH 7.4, 37°C, 100 microM forskolin, 10 mM NaF, 10 microM AlCl3 | Mus musculus | |
0.15 | - |
ATP | S49 cyc-, pH 7.4, 37°C, Mn2+, 100 microM forskolin | Mus musculus |
Metals/Ions | Comment | Organism | Structure |
---|---|---|---|
Mg2+ | - |
Mus musculus | |
Mn2+ | - |
Mus musculus |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Mus musculus | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
S49 cell | S49 lymphoma cell | Mus musculus | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP | - |
Mus musculus | cAMP + diphosphate | - |
? |
Synonyms | Comment | Organism |
---|---|---|
adenylyl cyclase | - |
Mus musculus |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.015 | - |
uridine 5'-(gamma-thio)triphosphate | S49 cyc-, Mn2+, 100 microM forskolin | Mus musculus | |
0.02 | - |
xanthosine 5'-(gamma-thio)triphosphate | S49 cyc-, Mn2+, 100 microM forskolin | Mus musculus | |
0.02 | - |
inosine 5'-(gamma-thio)triphosphate | Sf9, Mn2+, 100 microM forskolin, 10 mM NaF, 10 microM AlCl3 | Mus musculus | |
0.021 | - |
inosine 5'-(gamma-thio)triphosphate | S49 cyc-, Mn2+, 100 microM forskolin | Mus musculus | |
0.025 | - |
xanthosine 5'-(gamma-thio)triphosphate | Sf9, Mn2+, 100 microM forskolin, 10 mM NaF, 10 microM AlCl3 | Mus musculus | |
0.033 | - |
cytidine 5'-(gamma-thio)triphosphate | Sf9, Mn2+, 100 microM forskolin, 10 mM NaF, 10 microM AlCl3 | Mus musculus | |
0.051 | - |
uridine 5'-(gamma-thio)triphosphate | Sf9, Mn2+, 100 microM forskolin, 10 mM NaF, 10 microM AlCl3 | Mus musculus | |
0.071 | - |
cytidine 5'-(gamma-thio)triphosphate | S49 cyc-, Mn2+, 100 microM forskolin | Mus musculus | |
0.35 | - |
inosine 5'-(beta,gamma-imido)triphosphate | S49 cyc-, Mn2+, 100 microM forskolin | Mus musculus | |
0.4 | - |
guanosine 5'-(gamma-thio)triphosphate | Sf9, Mn2+, 100 microM forskolin, 10 mM NaF, 10 microM AlCl3 | Mus musculus | |
0.41 | - |
guanosine 5'-(gamma-thio)triphosphate | S49 cyc-, Mn2+, 100 microM forskolin | Mus musculus | |
0.44 | - |
GTP | Sf9, Mn2+, 100 microM forskolin, 10 mM NaF, 10 microM AlCl3 | Mus musculus | |
0.48 | - |
inosine 5'-(beta,gamma-imido)triphosphate | Sf9, Mn2+, 100 microM forskolin, 10 mM NaF, 10 microM AlCl3 | Mus musculus | |
0.55 | - |
XTP | S49 cyc-, Mn2+, 100 microM forskolin | Mus musculus | |
0.6 | - |
ITP | S49 cyc-, Mn2+, 100 microM forskolin | Mus musculus | |
0.67 | - |
GTP | S49 cyc-, Mn2+, 100 microM forskolin | Mus musculus | |
0.95 | - |
XTP | Sf9, Mn2+, 100 microM forskolin, 10 mM NaF, 10 microM AlCl3 | Mus musculus | |
0.99 | - |
ITP | Sf9, Mn2+, 100 microM forskolin, 10 mM NaF, 10 microM AlCl3 | Mus musculus | |
1 | - |
CTP | S49 cyc-, Mn2+, 100 microM forskolin | Mus musculus | |
1.1 | - |
UTP | S49 cyc-, Mn2+, 100 microM forskolin | Mus musculus | |
2.2 | - |
UTP | Sf9, Mn2+, 100 microM forskolin, 10 mM NaF, 10 microM AlCl3 | Mus musculus | |
2.4 | - |
guanosine 5'-(beta,gamma-imido)triphosphate | Sf9, Mn2+, 100 microM forskolin, 10 mM NaF, 10 microM AlCl3 | Mus musculus | |
2.5 | - |
uridine 5'-(beta,gamma-imido)triphosphate | S49 cyc-, Mn2+, 100 microM forskolin | Mus musculus | |
2.8 | - |
uridine 5'-(beta,gamma-imido)triphosphate | Sf9, Mn2+, 100 microM forskolin, 10 mM NaF, 10 microM AlCl3 | Mus musculus | |
2.9 | - |
CTP | Sf9, Mn2+, 100 microM forskolin, 10 mM NaF, 10 microM AlCl3 | Mus musculus | |
3 | - |
guanosine 5'-(beta,gamma-imido)triphosphate | S49 cyc-, Mn2+, 100 microM forskolin | Mus musculus | |
10 | - |
xanthosine 5'-(beta,gamma-imido)triphosphate | S49 cyc-, Mn2+, 100 microM forskolin | Mus musculus | |
10 | - |
xanthosine 5'-(beta,gamma-imido)triphosphate | Sf9, Mn2+, 100 microM forskolin, 10 mM NaF, 10 microM AlCl3 | Mus musculus |