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Literature summary for 4.2.99.18 extracted from

  • Raffoul, J.J.; Banerjee, S.; Singh-Gupta, V.; Knoll, Z.E.; Fite, A.; Zhang, H.; Abrams, J.; Sarkar, F.H.; Hillman, G.G.
    Down-regulation of apurinic/apyrimidinic endonuclease 1/redox factor-1 expression by soy isoflavones enhances prostate cancer radiotherapy in vitro and in vivo (2007), Cancer Res., 67, 2141-2149.
    View publication on PubMed

Application

Application Comment Organism
medicine selective targeting of APE1/Ref-1 could enhance conventional cancer treatment such as radiotherapy Mus musculus
medicine selective targeting of APE1/Ref-1 could enhance conventional cancer treatment such as radiotherapy Homo sapiens

Inhibitors

Inhibitors Comment Organism Structure
isoflavones soy isoflavones decrease apurinic/apyrimidinic endonuclease 1/redox factor-1 expression Homo sapiens
isoflavones soy isoflavones decrease apurinic/apyrimidinic endonuclease 1/redox factor-1 expression Mus musculus

Localization

Localization Comment Organism GeneOntology No. Textmining
cytoplasm
-
Mus musculus 5737
-
cytoplasm
-
Homo sapiens 5737
-
nucleus
-
Mus musculus 5634
-
nucleus
-
Homo sapiens 5634
-

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-
Mus musculus
-
male nude mice, BALB/c nu/nu 5-6 weeks old
-

Source Tissue

Source Tissue Comment Organism Textmining
PC-3 cell human prostate cancer cell line Homo sapiens
-
prostate cancer cell
-
Mus musculus
-

Synonyms

Synonyms Comment Organism
APE1
-
Mus musculus
APE1
-
Homo sapiens
apurinic/apyrimidinic endonuclease 1
-
Mus musculus
apurinic/apyrimidinic endonuclease 1
-
Homo sapiens
DNA-(apurinic or apyrimidinic site) lyase
-
Mus musculus
DNA-(apurinic or apyrimidinic site) lyase
-
Homo sapiens