Inhibitors | Comment | Organism | Structure |
---|---|---|---|
(1R,2S)-(-)-ephedrine | - |
Homo sapiens | |
(alpha-D-glucopyranosylthio)gold | - |
Homo sapiens | |
(R)-2,10,11-trihydroxy-N-propyl-noraporphine | - |
Homo sapiens | |
(R)-2,10,11-trihydroxyaporphine | - |
Homo sapiens | |
(R)-apomorphine | - |
Homo sapiens | |
(R)-N-allylnorapomorphine | - |
Homo sapiens | |
(R)-propylnorapomorphine | - |
Homo sapiens | |
(S)-carbidopa | - |
Homo sapiens | |
1-phenyl-2,3,4,5-tetrahydro-1H-3-benzazepine-7,8-diol | - |
Homo sapiens | |
3,4-dihydroxyphenylacetic acid | - |
Homo sapiens | |
4-chloromercuribenzoic acid | - |
Homo sapiens | |
4-[(2-sulfanyl-1H-imidazol-1-yl)methyl]phenol | - |
Homo sapiens | |
5'-guanidinonaltrindole | - |
Homo sapiens | |
6-amino-6,7-dihydroxy-1,2,3,4-tetrahydronaphthalene | - |
Homo sapiens | |
6-hydroxy-DL-DOPA | - |
Homo sapiens | |
aurintricarboxylic acid | - |
Homo sapiens | |
caffeic acid | - |
Homo sapiens | |
cephapirin | - |
Homo sapiens | |
dephostatin | - |
Homo sapiens | |
dihydrexidine | - |
Homo sapiens | |
ebselen | - |
Homo sapiens | |
hispidin | - |
Homo sapiens | |
hydroquinone | - |
Homo sapiens | |
iodoacetamide | - |
Homo sapiens | |
methyl 3-hydroxy-DL-tyrosinate | - |
Homo sapiens | |
myricetin | - |
Homo sapiens | |
N-acetyldopamine | - |
Homo sapiens | |
nordihydroguaiaretic acid | - |
Homo sapiens | |
p-benzoquinone | - |
Homo sapiens | |
piceatannol | - |
Homo sapiens | |
PPNDS tetrasodium | - |
Homo sapiens | |
SCH202676 | - |
Homo sapiens | |
SKF-89626 | - |
Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
HEK-293 cell | - |
Homo sapiens | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
5-fluorocytosine + H2O | - |
Homo sapiens | 5-fluorouracil + NH3 | - |
? |
Synonyms | Comment | Organism |
---|---|---|
APOBEC3G | - |
Homo sapiens |
Temperature Optimum [°C] | Temperature Optimum Maximum [°C] | Comment | Organism |
---|---|---|---|
37 | - |
assay at | Homo sapiens |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
7.4 | - |
assay at | Homo sapiens |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.00013 | - |
pH 7.4, 37°C | Homo sapiens | 4-chloromercuribenzoic acid | |
0.00017 | - |
pH 7.4, 37°C | Homo sapiens | p-benzoquinone | |
0.00036 | - |
pH 7.4, 37°C | Homo sapiens | (alpha-D-glucopyranosylthio)gold | |
0.00043 | - |
pH 7.4, 37°C | Homo sapiens | dephostatin | |
0.00045 | - |
pH 7.4, 37°C | Homo sapiens | N-acetyldopamine | |
0.00049 | - |
pH 7.4, 37°C | Homo sapiens | aurintricarboxylic acid | |
0.00059 | - |
pH 7.4, 37°C | Homo sapiens | dihydrexidine | |
0.0007 | - |
pH 7.4, 37°C | Homo sapiens | 6-amino-6,7-dihydroxy-1,2,3,4-tetrahydronaphthalene | |
0.0013 | - |
pH 7.4, 37°C | Homo sapiens | (R)-apomorphine | |
0.0013 | - |
pH 7.4, 37°C | Homo sapiens | SKF-89626 | |
0.0013 | - |
pH 7.4, 37°C | Homo sapiens | (1R,2S)-(-)-ephedrine | |
0.0017 | - |
pH 7.4, 37°C | Homo sapiens | (R)-2,10,11-trihydroxyaporphine | |
0.0018 | - |
pH 7.4, 37°C | Homo sapiens | piceatannol | |
0.002 | - |
pH 7.4, 37°C | Homo sapiens | hispidin | |
0.0026 | - |
pH 7.4, 37°C | Homo sapiens | hydroquinone | |
0.0028 | - |
pH 7.4, 37°C | Homo sapiens | ebselen | |
0.0029 | - |
pH 7.4, 37°C | Homo sapiens | (R)-N-allylnorapomorphine | |
0.003 | - |
pH 7.4, 37°C | Homo sapiens | iodoacetamide | |
0.0034 | - |
pH 7.4, 37°C | Homo sapiens | myricetin | |
0.0035 | - |
pH 7.4, 37°C | Homo sapiens | 4-[(2-sulfanyl-1H-imidazol-1-yl)methyl]phenol | |
0.004 | - |
pH 7.4, 37°C | Homo sapiens | 6-hydroxy-DL-DOPA | |
0.0053 | - |
pH 7.4, 37°C | Homo sapiens | (S)-carbidopa | |
0.0056 | - |
pH 7.4, 37°C | Homo sapiens | PPNDS tetrasodium | |
0.006 | - |
pH 7.4, 37°C | Homo sapiens | (R)-propylnorapomorphine | |
0.0064 | - |
pH 7.4, 37°C | Homo sapiens | 5'-guanidinonaltrindole | |
0.0075 | - |
pH 7.4, 37°C | Homo sapiens | cephapirin | |
0.0088 | - |
pH 7.4, 37°C | Homo sapiens | nordihydroguaiaretic acid | |
0.0091 | - |
pH 7.4, 37°C | Homo sapiens | dephostatin | |
0.013 | - |
pH 7.4, 37°C | Homo sapiens | methyl 3-hydroxy-DL-tyrosinate | |
0.013 | - |
pH 7.4, 37°C | Homo sapiens | (R)-2,10,11-trihydroxy-N-propyl-noraporphine | |
0.019 | - |
pH 7.4, 37°C | Homo sapiens | 3,4-dihydroxyphenylacetic acid | |
0.027 | - |
pH 7.4, 37°C | Homo sapiens | 1-phenyl-2,3,4,5-tetrahydro-1H-3-benzazepine-7,8-diol | |
0.029 | - |
pH 7.4, 37°C | Homo sapiens | SCH202676 | |
0.085 | - |
pH 7.4, 37°C | Homo sapiens | caffeic acid |