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Literature summary for 3.5.3.15 extracted from

  • Fujisaki, M.; Sugawara, K.
    Properties of peptidylarginine deiminase from the epidermis of newborn rats (1981), J. Biochem., 89, 257-263.
    View publication on PubMed

Activating Compound

Activating Compound Comment Organism Structure
dithiothreitol enhances activity, maximal activation at 2 mM Rattus norvegicus

Inhibitors

Inhibitors Comment Organism Structure
monoiodoacetate
-
Rattus norvegicus
PCMB
-
Rattus norvegicus

Metals/Ions

Metals/Ions Comment Organism Structure
Ca2+ required Rattus norvegicus
Ca2+ maximal activity in presence of 8-10 mM CaCl2 Rattus norvegicus
Ca2+ 10 mM, 11% of the activity with Ca2+ Rattus norvegicus
Sr2+ 10 mM, 85% of the activity with Ca2+ Rattus norvegicus

Molecular Weight [Da]

Molecular Weight [Da] Molecular Weight Maximum [Da] Comment Organism
48000
-
gel filtration Rattus norvegicus

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
protein L-Arg + H2O Rattus norvegicus citrullyl residues in the membranous protein of horny cells of the epidermis of newborn rat are formed by the action of epidermal peptidylarginine deiminase ?
-
?

Organism

Organism UniProt Comment Textmining
Rattus norvegicus
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
epidermis
-
Rattus norvegicus
-

Specific Activity [micromol/min/mg]

Specific Activity Minimum [µmol/min/mg] Specific Activity Maximum [µmol/min/mg] Comment Organism
0.00077
-
-
Rattus norvegicus

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
benzoyl-Gly-L-Arg + H2O
-
Rattus norvegicus benzoyl-Gly-L-citrulline + NH3
-
ir
benzoyl-L-Arg + H2O
-
Rattus norvegicus benzoyl-L-citrulline + NH3
-
ir
benzoyl-L-Arg-NH2 + H2O
-
Rattus norvegicus benzoyl-L-citrullineamide + NH3
-
ir
L-Arg + H2O negligible action Rattus norvegicus L-citrulline + NH3
-
?
protein L-Arg + H2O citrullyl residues in the membranous protein of horny cells of the epidermis of newborn rat are formed by the action of epidermal peptidylarginine deiminase Rattus norvegicus ?
-
?

Temperature Optimum [°C]

Temperature Optimum [°C] Temperature Optimum Maximum [°C] Comment Organism
50
-
-
Rattus norvegicus

pH Optimum

pH Optimum Minimum pH Optimum Maximum Comment Organism
7.5
-
-
Rattus norvegicus