Inhibitors | Comment | Organism | Structure |
---|---|---|---|
edrophonium | activity is reduced to 64.1% and 30.7% at 0.1 and 0.5 mM. Edrophonium inhibits esterase activity and aryl acylamidase activity of acetylcholinesterase | Homo sapiens | |
additional information | gallamine selectively inhibits the esterase activity to 63.6% (0.1 mM) and 45.4% (0.5 mM), whereas the aryl acylamidase activity remains significantly unaltered in the presence of gallamine (0.1 mM: 105.2%. 0.5 mM: 107%) | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | P22303 | cf. EC 3.1.1.7 | - |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
SAOS-2 cell | - |
Homo sapiens | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
2-nitroacetanilide + H2O | - |
Homo sapiens | 2-nitroaniline + acetate | - |
? |
General Information | Comment | Organism |
---|---|---|
physiological function | aryl acylamidase activity of acetylcholinesterase is actively involved in the process of osteoblast differentiation and mineralization | Homo sapiens |