Inhibitors | Comment | Organism | Structure |
---|---|---|---|
bortezomib | slow-binding inhibitor, kinetic analysis | Homo sapiens | |
delanzomib | slow-binding inhibitor, kinetic analysis | Homo sapiens | |
ixazomib | slow-binding inhibitor, kinetic analysis | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
succinyl-Leu-Leu-Val-Tyr-7-amido-4-methylcoumarin + H2O | - |
Homo sapiens | succinyl-Leu-Leu-Val-Tyr + 7-amino-4-methylcoumarin | - |
? |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.0000014 | - |
delanzomib | pH 8.0, 30°C | Homo sapiens | |
0.0000016 | - |
bortezomib | pH 8.0, 30°C | Homo sapiens | |
0.0000049 | - |
ixazomib | pH 8.0, 30°C | Homo sapiens |