Inhibitors | Comment | Organism | Structure |
---|---|---|---|
batimastat | - |
Homo sapiens | |
GM6001 | - |
Homo sapiens | |
marimastat | - |
Homo sapiens | |
MMP inhibitor III | - |
Homo sapiens | |
MMP inhibitor V | - |
Homo sapiens | |
MMP-3 inhibitor VIII | - |
Homo sapiens | |
TAPI-0 | - |
Homo sapiens | |
TAPI-1 | - |
Homo sapiens | |
TAPI-2 | - |
Homo sapiens |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
insulin-like growth factor binding protein-3 + H2O | Homo sapiens | - |
? | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | O43184 | - |
- |
Purification (Comment) | Organism |
---|---|
anion exchange column chromatography and concanavalin A column chromatography | Homo sapiens |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
HEK-293-EBNA cell | - |
Homo sapiens | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
5-Fam-EFPIYDFLPAKKK-NH2 + H2O | - |
Homo sapiens | 5-Fam-EFPI + YDFLPAKKK-NH2 | - |
? | |
5-Fam-FFLAQA(homophenylalanine)RSK-NH2 + H2O | best substrate | Homo sapiens | 5-Fam-FFLAQA + (homophenylalanine)RSK-NH2 | - |
? | |
5-Fam-HADLAQA(homophenylalanine)RSK-NH2 + H2O | - |
Homo sapiens | 5-Fam-HADLAQA + (homophenylalanine)RSK-NH2 | - |
? | |
5-Fam-HALAQA(homophenylalanine)RSK-NH2 + H2O | - |
Homo sapiens | 5-Fam-HALAQA + (homophenylalanine)RSK-NH2 | - |
? | |
5-Fam-LAQA(homophenylalanine)RSK-NH2 + H2O | - |
Homo sapiens | 5-Fam-LAQA + (homophenylalanine)RSK-NH2 | - |
? | |
5-Fam-SAVSRLRAYLLPA-NH2 + H2O | - |
Homo sapiens | 5-Fam-SAVSRLR + AYLLPA-NH2 | - |
? | |
Dabcyl-LAQA(homophenylalanine)RSK(5-FAM)-NH2 + H2O | - |
Homo sapiens | Dabcyl-LAQA + (homophenylalanine)RSK(5-FAM)-NH2 | - |
? | |
insulin-like growth factor binding protein-3 + H2O | - |
Homo sapiens | ? | - |
? |
Synonyms | Comment | Organism |
---|---|---|
ADAM12 | - |
Homo sapiens |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.000025 | - |
with 5-Fam-HALAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C | Homo sapiens | batimastat | |
0.000028 | - |
with 5-Fam-FFLAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C | Homo sapiens | batimastat | |
0.00012 | - |
with 5-Fam-FFLAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C | Homo sapiens | MMP inhibitor V | |
0.00018 | - |
with 5-Fam-HALAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C | Homo sapiens | MMP inhibitor V | |
0.00035 | - |
with 5-Fam-HALAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C | Homo sapiens | TAPI-0 | |
0.0004 | - |
with 5-Fam-FFLAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C | Homo sapiens | TAPI-0 | |
0.00043 | - |
with 5-Fam-FFLAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C | Homo sapiens | marimastat | |
0.0006 | - |
with 5-Fam-HALAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C | Homo sapiens | MMP inhibitor III | |
0.00067 | - |
with 5-Fam-HALAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C | Homo sapiens | marimastat | |
0.001 | - |
with 5-Fam-FFLAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C | Homo sapiens | TAPI-1 | |
0.0011 | - |
with 5-Fam-FFLAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C | Homo sapiens | MMP inhibitor III | |
0.0011 | - |
with 5-Fam-HALAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C | Homo sapiens | GM6001 | |
0.0014 | - |
with 5-Fam-FFLAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C | Homo sapiens | TAPI-2 | |
0.0014 | - |
with 5-Fam-HALAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C | Homo sapiens | TAPI-1 | |
0.0015 | - |
with 5-Fam-HALAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C | Homo sapiens | MMP-3 inhibitor VIII | |
0.0018 | - |
with 5-Fam-HALAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C | Homo sapiens | TAPI-2 | |
0.0021 | - |
with 5-Fam-FFLAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C | Homo sapiens | GM6001 | |
0.0028 | - |
with 5-Fam-FFLAQA(homophenylalanine)RSK-NH2 as substrate, at pH 8.0 and 22°C | Homo sapiens | MMP-3 inhibitor VIII |