Inhibitors | Comment | Organism | Structure |
---|---|---|---|
tissue inhibitor of metalloproteinase TIMP-1 | - |
Homo sapiens | |
tissue inhibitor of metalloproteinase TIMP-2 | - |
Homo sapiens |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.000013 | - |
stromelysin1 | pH 7.5, 37°C, monomeric form | Homo sapiens | |
0.000025 | - |
stromelysin1 | pH 7.5, 37°C, dimeric form | Homo sapiens |
Molecular Weight [Da] | Molecular Weight Maximum [Da] | Comment | Organism |
---|---|---|---|
92000 | - |
monomeric form, SDS-PAGE | Homo sapiens |
210000 | - |
dimeric form, SDS-PAGE | Homo sapiens |
225000 | - |
Western blot | Homo sapiens |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
additional information | Homo sapiens | associated with degradation of the extracellular matrix in normal and pathological conditions | ? | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | P45452 | human | - |
Purification (Comment) | Organism |
---|---|
- |
Homo sapiens |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
(7-methoxycoumaryl-4yl)acetylPLGLA2pr(2,4-dinitrophenol)-AR-NH2 + H2O | - |
Homo sapiens | ? | - |
? | |
additional information | associated with degradation of the extracellular matrix in normal and pathological conditions | Homo sapiens | ? | - |
? | |
stromelysin 1 + H2O | - |
Homo sapiens | ? | - |
? | |
stromelysin1 + H2O | - |
Homo sapiens | ? | - |
? |
Subunits | Comment | Organism |
---|---|---|
dimer | - |
Homo sapiens |
monomer | - |
Homo sapiens |
Synonyms | Comment | Organism |
---|---|---|
matrix metalloproteinase-9 | - |
Homo sapiens |
Turnover Number Minimum [1/s] | Turnover Number Maximum [1/s] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.00041 | - |
stromelysin 1 | pH 7.5, 37°C, dimeric form | Homo sapiens | |
0.0019 | - |
stromelysin 1 | pH 7.5, 37°C, monomeric form | Homo sapiens | |
0.04 | 1.97 | (7-methoxycoumaryl-4yl)acetylPLGLA2pr(2,4-dinitrophenol)-AR-NH2 | pH 7.5, 37°C, dimeric form | Homo sapiens | |
2.72 | - |
(7-methoxycoumaryl-4yl)acetylPLGLA2pr(2,4-dinitrophenol)-AR-NH2 | pH 7.5, 37°C, monomeric form | Homo sapiens | |
3 | 6 | (7-methoxycoumaryl-4yl)acetylPLGLA2pr(2,4-dinitrophenol)-AR-NH2 | pH 7.5, 37°C, monomeric form | Homo sapiens | |
8.67 | - |
(7-methoxycoumaryl-4yl)acetylPLGLA2pr(2,4-dinitrophenol)-AR-NH2 | pH 7.5, 37°C, dimeric form | Homo sapiens |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.00000713 | - |
TIMP-1 | pH 7.5, 37°C, dimeric form | Homo sapiens | |
0.00000817 | - |
TIMP-1 | pH 7.5, 37°C, monomeric form | Homo sapiens | |
0.0000259 | - |
TIMP-2 | pH 7.5, 37°C, monomeric form | Homo sapiens | |
0.0000361 | - |
TIMP-2 | pH 7.5, 37°C, dimeric form | Homo sapiens |