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Literature summary for 3.4.24.34 extracted from

  • Gavuzzo, E.; Pochetti, G.; Mazza, F.; Gallina, C.; Gorini, B.; D'Alessio, S.; Pieper, M.; Tschesche, H.; Tucker, P.A.
    Two crystal structures of human neutrophil collagenase, one complexed with a primed- and the other with an unprimed-side inhibitor: implications for drug design (2000), J. Med. Chem., 43, 3377-3385.
    View publication on PubMed

Crystallization (Commentary)

Crystallization (Comment) Organism
in complex with a primed and an unprimed-side inhibitor, hanging-drop vapor diffusion, space group P2(1)2(1)2(1), cell dimensions a : 32.98 A, b : 68.67 A, c : 70.49 A Homo sapiens

Inhibitors

Inhibitors Comment Organism Structure
(R)-2-(biphenyl-4-ylsulfonyl)-1,2,3,4-tetrahydroisoquinolin-3-carboxylic acid
-
Homo sapiens

Organism

Organism UniProt Comment Textmining
Homo sapiens P22894 human
-

Purification (Commentary)

Purification (Comment) Organism
catalytic domain Homo sapiens

Synonyms

Synonyms Comment Organism
HNC
-
Homo sapiens
MMP-8
-
Homo sapiens