Literature summary for 3.4.24.24 extracted from

Ikejiri, M.; Bernardo, M.M.; Meroueh, S.O.; Brown, S.; Chang, M.; Fridman, R.; Mobashery, S.
Design, synthesis, and evaluation of a mechanism-based inhibitor for gelatinase A (2005), J. Org. Chem., 70, 5709-5712.

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Inhibitors

Inhibitors	Comment	Organism	Structure
2-(4-(4-[(2-thiiranylpropyl)sulfonyl]phenoxy)phenyl)acetic acid	selective inhibitor	Homo sapiens
methyl 2-(4-(4-[(2-thiiranylpropyl)-sulfonyl]phenoxy)phenyl)acetate	mechanism-based inhibitor, selective for enzyme	Homo sapiens

Organism

Organism	UniProt	Comment	Textmining
Homo sapiens	-	-	-

Ki Value [mM]

Ki Value [mM]	Ki Value maximum [mM]	Inhibitor	Comment	Organism	Structure
0.00005	-	methyl 2-(4-(4-[(2-thiiranylpropyl)-sulfonyl]phenoxy)phenyl)acetate	-	Homo sapiens
0.00046	-	2-(4-(4-[(2-thiiranylpropyl)sulfonyl]phenoxy)phenyl)acetic acid	-	Homo sapiens

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Release 2023.1 (January 2023)