Inhibitors | Comment | Organism | Structure |
---|---|---|---|
(-)-5-hydroxypluviatolide | 50% inhibition at 0.05 mM | Homo sapiens | |
(-)-haplomyrfolin | 50% inhibition at 0.1 mM | Homo sapiens | |
(-)-hinokinin | 50% inhibition at 0.1 mM | Homo sapiens | |
(-)-thujaplicatin-d3 | 50% inhibition at 0.08 mM | Homo sapiens | |
additional information | for lignans, dibenzylbutyryrolactone structure is essential for inhibitory effect | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
recombinant enzyme | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
(7-methoxycoumarin-4-yl)acetyl-L-Pro-L-Leu-Gly-L-Leu-[N3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl]-L-Ala-L-Arg-NH2 + H2O | MOCAc-PLGL(Dpa)AR | Homo sapiens | ? | - |
? |