Cloned (Comment) | Organism |
---|---|
- |
Homo sapiens |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
acetyl-AEVD-CHO | - |
Homo sapiens | |
acetyl-DEVD-CHO | - |
Homo sapiens | |
acetyl-IETD-CHO | - |
Homo sapiens | |
acetyl-WEHD-CHO | - |
Homo sapiens | |
acetyl-YVAD-CHO | - |
Homo sapiens | |
benzyloxycarbonyl-VAD-fluoromethylketone | t1/2 at 0.001 mM is 3.9 s | Homo sapiens | |
cowpox serpin CrmA | the Ki-value is below 2.3 nM | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.000048 | - |
acetyl-AEVD-CHO | pH 7.5, 25°C | Homo sapiens | |
0.00006 | - |
acetyl-DEVD-CHO | pH 7.5, 25°C | Homo sapiens | |
0.000108 | - |
acetyl-IETD-CHO | pH 7.5, 25°C | Homo sapiens | |
0.000508 | - |
acetyl-WEHD-CHO | pH 7.5, 25°C | Homo sapiens | |
0.00097 | - |
acetyl-YVAD-CHO | pH 7.5, 25°C | Homo sapiens |