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Literature summary for 3.4.22.61 extracted from

  • Garcia-Calvo, M.; Peterson, E.P.; Leiting, B.; Ruel, R.; Nicholson, D.W.; Thornberry, N.A.
    Inhibition of human caspases by peptide-based and macromolecular inhibitors (1998), J. Biol. Chem., 273, 32608-32613.
    View publication on PubMed
Search for more literature for 3.4.22.61

Cloned(Commentary)

Cloned (Comment) Organism
-
 Homo sapiens

Inhibitors

Inhibitors Comment Organism Structure
acetyl-AEVD-aldehyde
-
 Homo sapiens
acetyl-DEVD-aldehyde
-
 Homo sapiens
acetyl-IETD-aldehyde
-
 Homo sapiens
acetyl-WEHD-aldehyde
-
 Homo sapiens
acetyl-YVAD-aldehyde
-
 Homo sapiens
benzyloxycarbonyl-Val-Ala-Asp-fluoromethylketone t1/2 at 0.001 mM: 2.5 s Homo sapiens
cowpox serpin CrmA Ki below 0.34 nM Homo sapiens

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Ki Value [mM]

Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
0.00000092
-
 acetyl-DEVD-aldehyde pH 7.5, 25°C Homo sapiens
0.00000105
-
 acetyl-IETD-aldehyde pH 7.5, 25°C Homo sapiens
0.0000016
-
 acetyl-AEVD-aldehyde pH 7.5, 25°C Homo sapiens
0.0000211
-
 acetyl-WEHD-aldehyde pH 7.5, 25°C Homo sapiens
0.000352
-
 acetyl-YVAD-aldehyde pH 7.5, 25°C Homo sapiens