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Literature summary for 3.4.22.52 extracted from

  • Hu, H.; Li, X.; Li, Y.; Wang, L.; Mehta, S.; Feng, Q.; Chen, R.; Peng, T.
    Calpain-1 induces apoptosis in pulmonary microvascular endothelial cells under septic conditions (2009), Microvasc. Res., 78, 33-39.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
calpain inhibitor-III
-
Mus musculus
calpastatin
-
Mus musculus

Organism

Organism UniProt Comment Textmining
Mus musculus
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
pulmonary microvascular endothelial cell
-
Mus musculus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
N-succinyl-LLVY-7-amido-4-methylcoumarin + H2O
-
Mus musculus N-succinyl-LLVY + 7-amino-4-methylcoumarin
-
?

Expression

Organism Comment Expression
Mus musculus in cultured pulmonary microvascular endothelial cells, incubation with septic plasma stimulates calpain activation. Reactive oxygen species produced from NADPH oxidase stimulates calpain-1 activation up

General Information

General Information Comment Organism
physiological function calpain-1 induces apoptosis in pulmonary microvascular endothelial cells under septic conditions Mus musculus